Potential of Essential Oil-Based Anticholinesterase Insecticides against Anopheles Vectors: A Review

TA Rants'o, LL Koekemoer, JL Panayides, RL van Zyl - Molecules, 2022 - mdpi.com
The insect nervous system is critical for its functional integrity. The cholinergic system, of
which acetylcholinesterase (AChE) is a key enzyme, is essential to the Anopheles …

Anopheles metabolic proteins in malaria transmission, prevention and control: a review

EO Adedeji, OO Ogunlana, S Fatumo, T Beder… - Parasites & vectors, 2020 - Springer
The increasing resistance to currently available insecticides in the malaria vector,
Anopheles mosquitoes, hampers their use as an effective vector control strategy for the …

Luminescent peptide/lanthanide (III) complex conjugates with push–pull antennas: application to one-and two-photon microscopy imaging

JH Choi, G Fremy, T Charnay, N Fayad… - Inorganic …, 2022 - ACS Publications
Lanthanide (III)(Ln3+) complexes feature desirable luminescence properties for cell
microscopy imaging, but cytosolic delivery of Ln3+ complexes and their use for 2P imaging …

Enzyme Dynamics Determine the Potency and Selectivity of Inhibitors Targeting Disease-Transmitting Mosquitoes

R Kumari, C Lindgren, R Kumar, N Forsgren… - ACS Infectious …, 2024 - ACS Publications
Vector control of mosquitoes with insecticides is an important tool for preventing the spread
of mosquito-borne diseases including malaria, dengue, chikungunya, and Zika …

Protected amine-functional initiators for the synthesis of α-amine homo-and heterotelechelic poly (2-ethyl-2-oxazoline) s

ZAI Mazrad, M Lai, TP Davis, JA Nicolazzo… - Polymer …, 2022 - pubs.rsc.org
Polymers bearing amine moieties are highly valuable for their ability to conjugate and/or
complex a variety of molecules. However, their incorporation into synthetic macromolecules …

Synthesis, biological evaluation, and computational investigation of ethyl 2, 4, 6-trisubstituted-1, 4-dihydropyrimidine-5-carboxylates as potential larvicidal agents …

R Duraisamy, NA Al-Shar'i… - Journal of …, 2024 - Taylor & Francis
Malaria is one of the most known vector-borne diseases caused by female Anopheles
mosquito bites. According to WHO, about 247 million cases of malaria and 619,000 deaths …

Larvicidal Activities of 2-Aryl-2,3-Dihydroquinazolin -4-ones against Malaria Vector Anopheles arabiensis, In Silico ADMET Prediction and Molecular Target …

KN Venugopala, P Ramachandra, C Tratrat… - Molecules, 2020 - mdpi.com
Malaria, affecting all continents, remains one of the life-threatening diseases introduced by
parasites that are transmitted to humans through the bites of infected Anopheles …

Sustainable use of plastic-derived nanocarbons as a promising larvicidal and growth inhibitor agent towards control of mosquitoes

V Shaw, R Koley, S Das, T Saha, NK Mondal - Science of The Total …, 2024 - Elsevier
Nanoscale carbon was obtained from six widely used plastics (PET, HDPE, PVC, LDPE, PP
and PP) via thermal degradation (600° C) under inert atmosphere. The thermally degraded …

Identification of a Novel Inhibitor of Cimex lectularius Acetylcholinesterase

J Qin, Z Yuchi - Journal of Agricultural and Food Chemistry, 2024 - ACS Publications
Acetylcholinesterase (AChE) stands as a primary target of commercial insecticides, notably
organophosphates and carbamates. Despite their widespread use in agricultural and indoor …

Broad‐Spectrum Antidote Discovery by Untangling the Reactivation Mechanism of Nerve‐Agent‐Inhibited Acetylcholinesterase

C Lindgren, N Forsgren, N Hoster… - … A European Journal, 2022 - Wiley Online Library
Reactivators are vital for the treatment of organophosphorus nerve agent (OPNA)
intoxication but new alternatives are needed due to their limited clinical applicability. The …