An update on the stereoselective synthesis of α-aminophosphonic acids and derivatives

M Ordonez, JL Viveros-Ceballos, C Cativiela… - Tetrahedron, 2015 - Elsevier
Optically active α-aminoalkylphosphonic acids 1 are structural analogues of α-amino acids
2, obtained by isosteric substitution of the planar and less bulky carboxylic acid (CO 2 H) by …

α‐Iminophosphonates: useful intermediates for enantioselective synthesis of α‐aminophosphonates

A Maestro, EM de Marigorta… - Asian Journal of …, 2020 - Wiley Online Library
A wide range of methods for the enantioselective synthesis of α‐aminophosphonic acid
derivatives have been developed over the years. Although the most used methodology is …

Synthesis, antioxidant and anticholinesterase activities of novel quinoline‐aminophosphonate derivatives

I Bazine, Z Cheraiet, R Bensegueni… - Journal of …, 2020 - Wiley Online Library
A series of 20 novel α‐aminophosphonate derivatives bearing quinoline or quinolone
moiety was designed and synthesized via Kabachnik‐Fields reaction in the presence of …

Highly efficient one-pot multi-component synthesis of α-aminophosphonates and bis-α-aminophosphonates catalyzed by heterogeneous reusable silica supported …

SAR Mulla, MY Pathan, SS Chavan, SP Gample… - RSC Advances, 2014 - pubs.rsc.org
A highly efficient one-pot multi-component reaction (MCR) protocol over DTP/SiO2 has been
developed for the synthesis of α-aminophosphonate derivatives (4a–x) in excellent yields …

[HTML][HTML] Synthesis of Novel 1,3,4-Oxadiazole-Derived α-Aminophosphonates/α-Aminophosphonic Acids and Evaluation of Their In Vitro Antiviral Activity against the …

S Hkiri, M Mekni-Toujani, E Üstün, K Hosni, A Ghram… - Pharmaceutics, 2022 - mdpi.com
An efficient and simple approach has been developed for the synthesis of eight dialkyl/aryl
[(5-phenyl-1, 3, 4-oxadiazol-2-ylamino)(aryl) methyl] phosphonates through the Pudovik …

[HTML][HTML] Silver(I) Complexes Based on Oxadiazole-Functionalized α-Aminophosphonate: Synthesis, Structural Study, and Biological Activities

S Hkiri, KA Coşkun, E Üstün, A Samarat, Y Tutar… - Molecules, 2022 - mdpi.com
Two silver (I) complexes, bis {diethyl [(5-phenyl-1, 3, 4-oxadiazol-2-yl-κ N 3: κ N 4-amino)(4-
trifluoromethylphenyl) methyl] phosphonate-(tetrafluoroborato-κ F)}-di-silver (I) and tetrakis …

Copper (II)-β-Cyclodextrin Promoted Kabachnik-Fields Reaction: An Efficient, One-Pot Synthesis of α-Aminophosphonates

R Keri, M Patil, VP Brahmkhatri, S Budagumpi… - Topics in …, 2022 - Springer
The design and application of environmental-friendly catalysts to reduce the toxic wastes are
critical for improving the chemical synthesis. Therefore, copper (II)-β-cyclodextrin catalyst …

Green synthesis, molecular docking, anti-oxidant and anti-inflammatory activities of α-aminophosphonates

M Sudileti, V Chintha, S Nagaripati, M Gundluru… - Medicinal Chemistry …, 2019 - Springer
The naturally viable α-amino acid surrogates have been synthesised via Kabachnik–Fields
reaction by the condensation of 2-aminothiazole with various aldehydes and dialkyl …

Potential antibacterial and antifungal activities of novel sulfamidophosphonate derivatives bearing the quinoline or quinolone moiety

I Bazine, S Bendjedid, A Boukhari - Archiv der Pharmazie, 2021 - Wiley Online Library
A series of new α‐sulfamidophosphonate/sulfonamidophosphonate (4a–n) and
cyclosulfamidophosphonate (5a–d) derivatives containing the quinoline or quinolone moiety …

Synthesis of α-aminophosphonates by the Kabachnik-Fields reaction

G Sravya, A Balakrishna, GV Zyryanov… - … , Sulfur, and Silicon …, 2020 - Taylor & Francis
The review discusses recent achievements in the development of more ecofriendly and
economically viable processes for the synthesis of biologically potent α-aminophosphonates …