The prevalence of nitrogen containing heterocycles in natural products and pharmaceuticals
is a doubtless fact. In this review, recent applications of a stereoselective aza-Michael …

Pyrroles are among the most privileged and influential small N-heterocycles at the core of
many commercial drugs, biological composition, natural compounds, agrochemicals, and …

A novel protocol for the preparation of functionalized 9-azabicyclo [3.3. 1] nonane (ABCN)
derivatives from 3-formylchromones, enaminones, and heterocyclic ketene aminals (HKAs) …

In contrast to the well‐established [3+ 2] cycloaddition reactions, the catalytic
enantioselective [3+ n](n≥ 3) cycloaddition reaction of activated isocyanides for the …

A novel protocol for the construction of highly functionalized bipyrimidine derivatives 4 and 5
from 3-formyl-chromones, ethyl 2-(pyridine-2-yl) acetate derivatives, and amidine …

We report herein an unprecedented atroposelective dynamic kinetic resolution of
Bringmann's lactones with C-nucleophiles. By the use of activated isocyanides as the …

The catalytic reaction of biaryl lactams with activated isocyanides is reported for the first time.
By employing a cooperative catalytic system, oxazole-containing axially chiral biaryl anilines …

A novel protocol was developed for preparing functionalized chromeno [2, 3-b] pyrrol-4 (1H)-
ones 3 (CMPOs) from 3-formylchromones with N-substituted glycine derivatives. The method …

An efficient and concise one-pot procedure was developed based on a cascade reaction of
3-formylchromones 1 and different types of 1, 1-enediamines (EDAMs) 2 with different …

A concise and efficient one-pot synthesis of novel N-fused tricyclic derivatives has been
developed by using the Groebke–Blackburn–Bienaymé (GBB) reaction, which involved the …