Potential nitrogen-based heterocyclic compounds for treating infectious diseases: a literature review

M Aatif, MA Raza, K Javed, SM Nashre-ul-Islam… - Antibiotics, 2022 - mdpi.com
Heterocyclic compounds are considered as one of the major and most diverse family of
organic compounds. Nowadays, the demand for these compounds is increasing day-by-day …

A comprehensive review on biological activities of oxazole derivatives

S Kakkar, B Narasimhan - BMC chemistry, 2019 - Springer
The utility of oxazole as intermediates for the synthesis of new chemical entities in medicinal
chemistry have been increased in the past few years. Oxazole is an important heterocyclic …

Development of newly synthesised quinazolinone-based CDK2 inhibitors with potent efficacy against melanoma

ER Mohammed, GF Elmasry - Journal of Enzyme Inhibition and …, 2022 - Taylor & Francis
Inhibiting Cyclin-dependent kinase 2 (CDK2) has been established as a therapeutic strategy
for the treatment of many cancers. Accordingly, this study aimed at developing a new set of …

Synthesis, characterization, theoretical studies, and antimicrobial/antitumor potencies of salen and salen/imidazole complexes of Co (II), Ni (II), Cu (II), Cd (II), Al (III) …

EM Abdalla, LH Abdel Rahman… - Applied …, 2020 - Wiley Online Library
Although salens and imidazoles are well‐studied motifs among bioactive and therapeutic
agents, their properties when combined in transition metal complexes are not well …

Microwave Assisted Improved Method for the Synthesis of Pyrazole Containing 2, 4,‐Disubstituted Oxazole‐5‐one and their Antimicrobial Activity

ND Argade, BK Kalrale, CH Gill - Journal of Chemistry, 2008 - Wiley Online Library
Disubstituted oxazol‐5‐one and pyrazoles are known to exhibit various biological activities.
Therefore, in this work, we designed pyrazole containing 2, 4‐disubstituted oxazol‐5‐one …

5(4H)-oxazolones: Synthesis and biological activities

DSA Haneen, WSI Abou-Elmagd… - Synthetic …, 2021 - Taylor & Francis
Full article: 5(4H)-oxazolones: Synthesis and biological activities Skip to Main Content Taylor and
Francis Online homepage Taylor and Francis Online homepage Log in | Register Cart 1.Home 2.All …

Exploring new quinazolin‐4(3H)‐one derivatives as CDK2 inhibitors: Design, synthesis, and anticancer evaluation

BT Ibrahim, HA Allam, NM El‐Dydamony… - Drug Development …, 2024 - Wiley Online Library
In the present work, five series of new 2, 3‐disubstituted quinazolin‐4 (3H)‐ones 4a–c, 5a–
d, 6a–g, 7a, b, and 9a–c were designed, synthesized, and screened in vitro for their cytotoxic …

Nano Fe2O3, clinoptilolite and H3PW12O40 as efficient catalysts for solvent-free synthesis of 5 (4H)-isoxazolone under microwave irradiation conditions

S Fozooni, NG Hosseinzadeh, H Hamidian… - Journal of the Brazilian …, 2013 - SciELO Brasil
A quick and solvent-free approach involving the exposure of neat reactants to microwave
irradiation in conjunction with the use of clinoptilolite, H3PW12O40 and Fe2O3 nanoparticle …

Preparation and characterization of supported bimetallic gold–iron nanoparticles, and its potential for heterogeneous catalysis

G Ferouani, N Ameur, R Bachir - Research on Chemical Intermediates, 2020 - Springer
Bimetallic gold–iron catalysts supported on ZrO 2 and TiO 2 were prepared by under
potential deposition. The characterization of the catalysts was performed using an …

[HTML][HTML] Synthesis and antitumor activity of certain 2, 3, 6-trisubstituted quinazolin-4 (3H)-one derivatives

SE Abbas, FF Barsoum, HH Georgey… - Bulletin of Faculty of …, 2013 - Elsevier
The synthesis of different series of 6-iodo-2-phenoxymethyl 3-substituted quinazolin-4 (3H)-
ones 5–17 is described. The structures of the newly synthesized compounds have been …