Medicinal applications of coumarins bearing azetidinone and thiazolidinone moieties
Coumarins (2 H-chromen-2-ones), also known as benzopyran-2-ones, are a family of
naturally occurring heterocyclic ring systems that contain a lactone moiety. Coumarins …
naturally occurring heterocyclic ring systems that contain a lactone moiety. Coumarins …
Rational design and synthesis of new tetralin-sulfonamide derivatives as potent anti-diabetics and DPP-4 inhibitors: 2D & 3D QSAR, in vivo radiolabeling and bio …
SS Abd El-Karim, MM Anwar, YM Syam, MA Nael… - Bioorganic …, 2018 - Elsevier
Abstract Type 2 diabetes (T2D) is a severe disease and it is one of the most raising
problems worldwide. This study deals with design, synthesis and in vivo determination of a …
problems worldwide. This study deals with design, synthesis and in vivo determination of a …
[PDF][PDF] A BRIEF REVIEW ON RECENT SYNTHESIS OF 2-AZETIDINONE DERIVATIVES.
DS Salunkhe, PB Piste - International Journal of Pharmacy & Life …, 2014 - researchgate.net
The chemistry of β-lactams has taken an prestigious place in organic and medicinal
chemistry so the review on recent methods in the synthesis of 2-Azetidinone derivatives …
chemistry so the review on recent methods in the synthesis of 2-Azetidinone derivatives …
Synthesis and biological activity of novel hydantoin cyclohexyl sulfonamide derivatives as potential antimicrobial agents in agriculture
W Liu, S Zhang, L Xiao, Y Wan, L He… - Pest Management …, 2022 - Wiley Online Library
BACKGROUND Plant disease is one of the most serious problems in agriculture that can
damage crops. Chemical fungicides are widely used to control plant diseases, but have led …
damage crops. Chemical fungicides are widely used to control plant diseases, but have led …
[PDF][PDF] Synthesis, characterization and antibacterial activity of some new of novel 1, 2, 3-triazole-chalcone derivatives from N-acetyl-5H-dibenzo [B, F] azepine-5 …
This work involves preparation of a series of 1, 2, 3-triazole derivatives. In the first step, the
reaction of N-acetyl-5H-dibenzo [b, f] carboxamide with different benzaldehyde derivatives to …
reaction of N-acetyl-5H-dibenzo [b, f] carboxamide with different benzaldehyde derivatives to …
[PDF][PDF] Synthesis and discerning of antibiotic potential of PCMX based novel azetidinones
Azetidinones and PCMX are potent antimicrobial entities. The cyclocondensation of N-
substituted benzylidene-2-(4-chloro-3, 5-dimethylphenoxy) acetamide (2a-e), with TEA and …
substituted benzylidene-2-(4-chloro-3, 5-dimethylphenoxy) acetamide (2a-e), with TEA and …
Visible light-induced degradation of sulfa drugs on pure TiO2 through ligand-to-metal charge transfer
The degradation of sulfisoxazole (SSX) on pure TiO 2 under visible light irradiation was
investigated. 50 µM SSX was completely degraded in a suspension of pure TiO 2 (Hombikat …
investigated. 50 µM SSX was completely degraded in a suspension of pure TiO 2 (Hombikat …
Development and characterization of novel films based on sulfonamide-chitosan derivatives for potential wound dressing
OM Dragostin, SK Samal, F Lupascu… - International Journal of …, 2015 - mdpi.com
The objective of this study was to develop new films based on chitosan functionalized with
sulfonamide drugs (sulfametoxydiazine, sulfadiazine, sulfadimetho-xine, sulfamethoxazol …
sulfonamide drugs (sulfametoxydiazine, sulfadiazine, sulfadimetho-xine, sulfamethoxazol …
[PDF][PDF] New arginine derivatives-synthesis and biological evaluation
A Pânzariu, IM Vasincu, OM Dragostin, M Drăgan… - Farmacia, 2015 - researchgate.net
A novel series of L-arginine derivates with imine structure (Schiff bases) were synthetized
and the structure was confirmed using spectral methods: infrared (IR), nuclear magnetic …
and the structure was confirmed using spectral methods: infrared (IR), nuclear magnetic …
N-(4-取代氨基磺酰基) 苯基-酮基蒎酸酰胺的合成及生物活性
吴光燧, 段文贵, 林桂汕, 岑波, 赵莉, 雷福厚 - 农药学学报, 2014 - nyxxb.cn
以D-(+)-樟脑磺酸为原料, 经酰氯化和氧化反应制备得到酮基蒎酸(3), 再经酰氯化得到酮基蒎酸
酰氯(4). 4 与对氨基苯磺酰胺类化合物发生N-酰化反应, 得到8 个未见文献报道的N-(4 …
酰氯(4). 4 与对氨基苯磺酰胺类化合物发生N-酰化反应, 得到8 个未见文献报道的N-(4 …