Recent developments in azole compounds as antibacterial and antifungal agents

XM Peng, GX Cai, CH Zhou - Current Topics in Medicinal …, 2013 - ingentaconnect.com
Azole compounds are an important class of nitrogen heterocycles with electron-rich
property. This special structure endows azole-based derivatives easily bind with the …

[PDF][PDF] Antibacterial activity of thiazole and its derivatives

P Mohanty, S Behera, R Behura… - … Res. Appl. Chem, 2021 - biointerfaceresearch.com
Thiazoles are one of the most intensively scrutinized classes of 5-membered aromatic
heterocycles. Many natural and synthesized thiazole and its derivatives showed significant …

1, 2, 3-Triazole derivatives as antitubercular agents: synthesis, biological evaluation and molecular docking study

MH Shaikh, DD Subhedar, L Nawale, D Sarkar… - …, 2015 - pubs.rsc.org
Searching for new active molecules against Mycobacterium tuberculosis (MTB) H37Ra, a
small focused library of 1, 2, 3-triazoles has been efficiently prepared via a click chemistry …

Synthesis and bioactivity of novel triazole incorporated benzothiazinone derivatives as antitubercular and antioxidant agent

MH Shaikh, DD Subhedar, M Arkile, VM Khedkar… - Bioorganic & medicinal …, 2016 - Elsevier
In search of new active molecules against Mycobacterium tuberculosis (MTB) H37Ra and M.
bovis BCG, a small focused library of benzothiazinone based 1, 2, 3-triazoles has been …

Synthesis, biological evaluation and molecular docking of novel coumarin incorporated triazoles as antitubercular, antioxidant and antimicrobial agents

MH Shaikh, DD Subhedar, BB Shingate… - Medicinal Chemistry …, 2016 - Springer
A series of new coumarin-based 1, 2, 3-triazole derivatives were designed, synthesized and
evaluated for their antitubercular activity in vitro against Mycobacterium tuberculosis H37Ra …

1, 2, 3-Triazole incorporated coumarin derivatives as potential antifungal and antioxidant agents

MH Shaikh, DD Subhedar, FAK Khan… - Chinese Chemical …, 2016 - Elsevier
A series of novel ethyl-7-((1-(benzyl)-1H-1, 2, 3-triazol-4-yl) methoxy)-2-oxo-2H-chromene-3-
carboxylates 8a-h as potential antifungal agents were synthesized via click chemistry. The …

Facile one-pot multicomponent synthesis and molecular docking studies of steroidal oxazole/thiazole derivatives with effective antimicrobial, antibiofilm and hemolytic …

A Ansari, A Ali, M Asif, MA Rauf, M Owais - Steroids, 2018 - Elsevier
A series of steroidal oxazole and thiazole derivatives have been synthesized employing
thiosemicarbazide/semicarbazide hydrochloride and ethyl 2-chloroacetoacetate with a …

Novel tetrazoloquinoline–rhodanine conjugates: highly efficient synthesis and biological evaluation

DD Subhedar, MH Shaikh, L Nawale, A Yeware… - Bioorganic & Medicinal …, 2016 - Elsevier
In search of new active molecules against Mycobacterium tuberculosis (MTB) H37Ra and
Mycobacterium bovis BCG, a small focused library of rhodanine incorporated …

Novel alkylaminoethyl derivatives of androstane 3-oximes as anticancer candidates: Synthesis and evaluation of cytotoxic effects

JJ Ajduković, DS Jakimov, L Rárová, M Strnad… - RSC …, 2021 - pubs.rsc.org
Steroid anticancer drugs are the focus of numerous scientific research efforts. Due to their
high cytotoxic effects against tumor cells, some natural or synthetic steroid compounds seem …

[Et3NH][HSO4] catalyzed efficient synthesis of 5-arylidene-rhodanine conjugates and their antitubercular activity

DD Subhedar, MH Shaikh, L Nawale, A Yeware… - Research on chemical …, 2016 - Springer
We have described a highly efficient, safer protocol for the synthesis of 5-arylidene-
rhodanine conjugates catalyzed by Bronsted acidic ionic liquid [Et 3 NH][HSO 4] in excellent …