Discovery of 9H-pyrimido [4, 5-b] indole derivatives as dual RET/TRKA inhibitors

B Acharya, D Saha, NG Garcia, D Armstrong… - Bioorganic & Medicinal …, 2024 - Elsevier
Aberrant RET kinase signaling is activated in numerous cancers including lung, thyroid,
breast, pancreatic, and prostate. Recent approvals of selective RET inhibitors, pralsetinib …

[HTML][HTML] Tyrosine Kinase Inhibitors and Thyroid Toxicity

S Mastrangelo, G Attina… - Biomedical and …, 2023 - biomedpharmajournal.org
Some multithyrosine kinase inhibitors have been reported to cause changes in thyroid
function. For the management of sunitinib-induced hypothyroidism, an evaluation of thyroid …