Hydration effects on molecular structure, vibrational, electronic properties, drug-likeness analysis, molecular docking, and molecular dynamics studies of (Z)-3-(2-oxo …

SJ Koyambo-Konzapa, SO Aljazzar… - Journal of Molecular …, 2024 - Elsevier
This study examines how solvation models, including COSMO, CPCM, PCM, and SMD,
affect the conformations, molecular structure, vibrational behaviors, and electronic properties …

Identification of diosmin and flavin adenine dinucleotide as repurposing treatments for monkeypox virus: a computational study

TP Lam, VH Tran, TT Mai, NVT Lai, BTN Dang… - International Journal of …, 2022 - mdpi.com
The World Health Organization declared monkeypox a global public health emergency on
23 July 2022. This disease was caused by the monkeypox virus (MPXV), which was first …

Acemannan ameliorates STZ-activated diabetes by attenuating high glucose via inhibiting inflammatory cytokines and apoptosis pathway

AB Omer, HN Altayb, FA Al-Abbasi, G Gupta… - International journal of …, 2023 - Elsevier
Acemannan, the main polysaccharide in Aloe vera, is a-(1, 4)-acetylated polymannose.
According to numerous research findings, acemannan is a viable alternative for the …

QSAR, Molecular Docking, and Dynamics-Based Computational discovery of Potential PLK4 Inhibitors for tumor therapy

Y Liu, JB Tong, X Fan - Process Biochemistry, 2024 - Elsevier
Abstract PLK4 (polo-like kinase 4), an enzyme regulating centrioles, has been identified as a
highly promising target for cancer treatment, making the development of PLK4 inhibitors …

Designing of 2, 3-dihydrobenzofuran derivatives as inhibitors of PDE1B using pharmacophore screening, ensemble docking and molecular dynamics approach

M Al-Nema, A Gaurav, VS Lee - Computers in Biology and Medicine, 2023 - Elsevier
In recent years, the PDE1B enzyme has become a desirable drug target for the treatment of
psychological and neurological disorders, particularly schizophrenia disorder, due to the …

In silico molecular docking and dynamic simulation of anti-cholinesterase compounds from the extract of Catunaregam spinosa for possible treatment of Alzheimer's …

S Thandivel, P Rajan, T Gunasekar, A Arjunan, S Khute… - Heliyon, 2024 - cell.com
Abstract Alzheimer's disease (AD), is characterized by a progressive loss of cognitive
abilities as well as behavioral symptoms including disorientation, trouble solving problems …

[HTML][HTML] Molecular docking and dynamics simulation study of medicinal fungi derived secondary metabolites as potential inhibitor for COVID-19 treatment

MAS Khan, MI Miah, Z Islam, S Afrin, MF Ahmed… - Informatics in Medicine …, 2023 - Elsevier
The severity of COVID-19, lack of specific treatment, and controversies on the vaccine's
efficacy demand the development of new drugs against SARS-CoV-2. Fungi produce …

Phytochemical Screening of Ultrasonic Extracts of Salix Species and Molecular Docking Study of Salix-Derived Bioactive Compounds Targeting Pro-Inflammatory …

E Gligorić, R Igić, B Teofilović… - International Journal of …, 2023 - mdpi.com
Willow bark (Salix spp., Salicaceae) is a traditional analgesic and antirheumatic herbal
medicine. The aim of this study was to evaluate and compare the phytochemical and …

In Silico Molecular Docking and Dynamic Investigations of Bioactive Phytoconstituents from Fenugreek Seeds as a Potent Drug against DPP-IV Enzyme

DK Sarker, P Ray, R Rouf, JA Shilpi… - ACS Food Science & …, 2023 - ACS Publications
Type 2 diabetes is a metabolic disorder resulting from impaired insulin action or dysfunction
in β cells. The incretin hormone, glucagon-like peptide-1, is secreted during the meal intake …

In silico approach to identify novel allosteric intracellular antagonist for blocking the interleukin-8/CXCR2 receptor signaling pathway

TTN Tran, QH Tran, CQ Duong… - Journal of …, 2023 - Taylor & Francis
The role of interleukin-8 (IL-8) and its receptor CXCR2 in inflammatory responses and tumor
development and progression has been well documented. Our study aims to discover novel …