Substituted [1, 2, 4] triazolo [1, 5-a] pyrazines as LSD1 inhibitors
L Wu, X Wang, W Yao, C Zhang - US Patent 10,968,221, 2021 - Google Patents
Int. Ci. A61K 31/4985 (2006.01) CO7D 487/04 (2006.01) C070 471/04(2006.01)(52) US
CI.??? CO7D 471/04 (2013.01); C07D 487704 (2013.01)(58) Field of Classification Search …
CI.??? CO7D 471/04 (2013.01); C07D 487704 (2013.01)(58) Field of Classification Search …
Salts of an LSD1 inhibitor and processes for preparing the same
Z Jia, W Han, Y Pan, T Martin, J Zhou, Q Li - US Patent 10,968,200, 2021 - Google Patents
(57) ABSTRACT 4,537,889 A 4,625,040 A 5,658,857 A 5,932,223 A 7,759,386 B2 7,858,609
B2 8,115,000 B2 8,349,210 B2 8,383,154 B2 8,546,394 B2 8,558,008 B2 8,568,782 B2 …
B2 8,115,000 B2 8,349,210 B2 8,383,154 B2 8,546,394 B2 8,558,008 B2 8,568,782 B2 …
Fused pyrimidine derivatives as A2A/A2B inhibitors
X Wang, H Han, MS McCammant, L Wu… - US Patent …, 2021 - Google Patents
8,288,536 B2 8,349,850 B2 8,431,596 B2 8,569,300 B2 8,575,183 B2 8,580,812 B2
8,637,542 B2 8,865,731 B2 8,865,734 B2 9,029,389 B2 9,029,393 B2 9,034,872 B2 …
8,637,542 B2 8,865,731 B2 8,865,734 B2 9,029,389 B2 9,029,393 B2 9,034,872 B2 …
Imidazopyrimidines and triazolopyrimidines as a2a/a2b inhibitors
X Wang, P Gan, T Huang, C Qi, DQ Qian, L Wu… - US Patent …, 2023 - Google Patents
2022-05-12 Assigned to INCYTE CORPORATION reassignment INCYTE CORPORATION
ASSIGNMENT OF ASSIGNORS INTEREST (SEE DOCUMENT FOR DETAILS). Assignors …
ASSIGNMENT OF ASSIGNORS INTEREST (SEE DOCUMENT FOR DETAILS). Assignors …
Pyrazolopyridines and triazolopyridines as A2A/A2B inhibitors
T Huang, X Wang - US Patent 11,390,624, 2022 - Google Patents
6,545,000 B1 6,921,762 B2 7,041,666 B2 7,306,631 B2 7,452,892 B2 7,501,411 B2
7,511,050 B2 7,563,788 B2 7,674,791 B2 7,700,594 B2 7,709,468 B2 7,834,014 B2 …
7,511,050 B2 7,563,788 B2 7,674,791 B2 7,700,594 B2 7,709,468 B2 7,834,014 B2 …
Salts of an LSD1 inhibitor
Y Pan, W Han, G Cao, Z Jia, J Zhou - US Patent 11,498,900, 2022 - Google Patents
The present disclosure relates to tosylate salts 1-{[4 (methoxymethyl)-4-({[(1R, 2S)-2-
phenylcyclopropyl] amino} methyl) piperidin-1-yl] methyl} cyclobutanecarboxylic acid …
phenylcyclopropyl] amino} methyl) piperidin-1-yl] methyl} cyclobutanecarboxylic acid …
Cyclopropylamines as LSD1 inhibitors
L Wu, JR Courter, C He, X Wang, W Yao… - US Patent …, 2022 - Google Patents
First worldwide family litigation filed litigation Critical https://patents. darts-ip. com/? family=
52589819&utm_source= google_patent&utm_medium= platform_link&utm_campaign …
52589819&utm_source= google_patent&utm_medium= platform_link&utm_campaign …
Cyclopropylamines as LSD1 inhibitors
L Wu, W Yao - US Patent 11,155,532, 2021 - Google Patents
4,537,889 A 4,625,040 A 5,658,857 A 5,932,223 A 7,759,386 B2 7,858,609 B2 8,115,000
B2 8,349,210 B2 8,383,154 B2 8,546,394 B2 8,558,008 B2 8,568,782 B2 8,614,315 B2 …
B2 8,349,210 B2 8,383,154 B2 8,546,394 B2 8,558,008 B2 8,568,782 B2 8,614,315 B2 …
Salts of an LSD1 inhibitor and processes for preparing the same
Z Jia, W Han, Y Pan, T Martin, J Zhou, Q Li - US Patent 11,512,064, 2022 - Google Patents
NOGBPURWUNSIIC-GGYWPGCISA-N N# CCC1 (N2CCC (CC3C [C@ H] 3c3ccccc3) CC2)
CN (S (N)(= O)= O) C1 Chemical compound N# CCC1 (N2CCC (CC3C [C@ H] 3c3ccccc3) …
CN (S (N)(= O)= O) C1 Chemical compound N# CCC1 (N2CCC (CC3C [C@ H] 3c3ccccc3) …
Pyrazolopyridines and triazolopyridines as A2A/A2B inhibitors
T Huang, X Wang - US Patent 11,884,665, 2024 - Google Patents
MSXIFXOIITVIOS-UHFFFAOYSA-N 3-[4-amino-2-[(3-fluoropyridin-2-yl) methyl]-7-pyrimidin-4-
yltriazolo [4, 5-c] pyridin-6-yl] benzonitrile Chemical compound NC1= NC (= C (C= 2C1= NN …
yltriazolo [4, 5-c] pyridin-6-yl] benzonitrile Chemical compound NC1= NC (= C (C= 2C1= NN …