Nanocrystals as a master key to deliver hydrophobic drugs via multiple administration routes

MB McGuckin, J Wang, R Ghanma, N Qin… - Journal of Controlled …, 2022 - Elsevier
The poor aqueous solubility of many approved drugs and most new chemical entities poses
a challenge to drug delivery scientists working in academic and industrial labs. Despite the …

Long-acting injectable antiretrovirals for HIV treatment and prevention

WR Spreen, DA Margolis… - Current Opinion in HIV …, 2013 - journals.lww.com
Investigational long-acting injectable nanoformulations of rilpivirine and GSK1265744 are
clinical-stage development candidates. Complementary pharmacologic properties of both …

Atazanavir, alone or in combination with ritonavir, inhibits SARS-CoV-2 replication and proinflammatory cytokine production

N Fintelman-Rodrigues, CQ Sacramento… - Antimicrobial agents …, 2020 - Am Soc Microbiol
Severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2) is already responsible for
far more deaths than previous pathogenic coronaviruses (CoVs) from 2002 and 2012. The …

Long-acting HIV drugs for treatment and prevention

RM Gulick, C Flexner - Annual review of medicine, 2019 - annualreviews.org
Antiretroviral drugs have revolutionized the treatment and prevention of HIV infection;
however, adherence is critical for sustained efficacy. Current HIV treatment consists of three …

Creation of a long-acting nanoformulated dolutegravir

B Sillman, AN Bade, PK Dash, B Bhargavan… - Nature …, 2018 - nature.com
Potent antiretroviral activities and a barrier to viral resistance characterize the human
immunodeficiency virus type one (HIV-1) integrase strand transfer inhibitor dolutegravir …

Recent advances in long-acting nanoformulations for delivery of antiretroviral drugs

DH Surve, AB Jindal - Journal of Controlled Release, 2020 - Elsevier
In spite of introduction of combination antiretroviral therapy (cART) against human
immunodeficiency virus (HIV) infection; inaccessibility and poor adherence to oral cART …

Long-acting antiviral agents for HIV treatment

DA Margolis, M Boffito - Current Opinion in HIV and AIDS, 2015 - journals.lww.com
Phase II studies evaluating the coadministration of rilpivirine and cabotegravir
intramuscularly to HIV-infected individuals with an undetectable viral load are currently …

Development of HIV reservoir targeted long acting nanoformulated antiretroviral therapies

BJ Edagwa, T Zhou, JE M McMillan… - Current medicinal …, 2014 - ingentaconnect.com
Human immunodeficiency virus (HIV) infection commonly results in a myriad of comorbid
conditions secondary to immune deficiency. Infection also affects broad organ system …

Long-acting slow effective release antiretroviral therapy

B Edagwa, JE McMillan, B Sillman… - Expert opinion on drug …, 2017 - Taylor & Francis
Introduction: Advances in long-acting antiretroviral therapy (ART) can revolutionize current
HIV/AIDS treatments. We coined the term 'long-acting slow effective release ART'(LASER …

Dolutegravir, the second-generation of integrase strand transfer inhibitors (INSTIs) for the treatment of HIV

DE Dow, JA Bartlett - Infectious diseases and therapy, 2014 - Springer
The integrase strand transfer inhibitors (INSTIs) are the newest antiretroviral class in the HIV
treatment armamentarium. Dolutegravir (DTG) is the only second-generation INSTI with FDA …