Role of calixarene in chemotherapy delivery strategies
R Basilotta, D Mannino, A Filippone, G Casili… - Molecules, 2021 - mdpi.com
Since cancer is a multifactorial disease with a high mortality rate, the study of new
therapeutic strategies is one of the main objectives in modern research. Numerous …
therapeutic strategies is one of the main objectives in modern research. Numerous …
The Odd Couple (s): An overview of Beta-Lactam antibiotics bearing more than one pharmacophoric group
M De Rosa, A Verdino, A Soriente… - International Journal of …, 2021 - mdpi.com
β-lactam antibiotics are among the most important and widely used antimicrobials worldwide
and are comprised of a large family of compounds, obtained by chemical modifications of …
and are comprised of a large family of compounds, obtained by chemical modifications of …
Thiacalixarene based quaternary ammonium salts as promising antibacterial agents
PL Padnya, OS Terenteva, AA Akhmedov… - Bioorganic & Medicinal …, 2021 - Elsevier
The search for new antibacterial and antiseptic drugs is an urgent problem due to the
resistance of microorganisms to existing drugs. In this work, for the first time, the design of …
resistance of microorganisms to existing drugs. In this work, for the first time, the design of …
A novel material based on an antibacterial choline-calixarene nanoassembly embedded in thin films
L Ferreri, GML Consoli, G Clarizia, DC Zampino… - Journal of Materials …, 2022 - Springer
Supramolecular chemistry is one of the current strategies for producing advanced materials.
With the aim to develop new Thin-Films with antibacterial activity, we embedded an …
With the aim to develop new Thin-Films with antibacterial activity, we embedded an …
Peptidomimetics based on ammonium decasubstituted pillar [5] arenes: Influence of the alpha-amino acid residue nature on cholinesterase inhibition
Cholinesterase inhibitors are a group of medicines that are widely used for the treatment of
cognitive impairments accompanying Alzheimer's disease as well as for the treatment of …
cognitive impairments accompanying Alzheimer's disease as well as for the treatment of …
Bismacrocycle: Structures and Applications
XL Chen, SQ Yu, XH Huang, HY Gong - Molecules, 2023 - mdpi.com
In the past half-century, macrocycles with different structures and functions, have played a
critical role in supramolecular chemistry. Two macrocyclic moieties can be linked to form …
critical role in supramolecular chemistry. Two macrocyclic moieties can be linked to form …
PAMAM-calix-dendrimers: Synthesis and thiacalixarene conformation effect on DNA binding
A convenient method for the synthesis of the first generation PAMAM dendrimers based on
the thiacalix [4] arene has been developed for the first time. Three new PAMAM-calix …
the thiacalix [4] arene has been developed for the first time. Three new PAMAM-calix …
PAMAM-calix-dendrimers: Second generation synthesis, fluorescent properties and catecholamines binding
O Mostovaya, I Shiabiev, D Pysin, A Stanavaya… - Pharmaceutics, 2022 - mdpi.com
A convenient method for the synthesis of the second generation of PAMAM dendrimers
based on a p-tert-butylthiacalix [4] arene core in cone, partial cone and 1, 3-alternate …
based on a p-tert-butylthiacalix [4] arene core in cone, partial cone and 1, 3-alternate …
Self-healing thiolated pillar [5] arene films containing moxifloxacin suppress the development of bacterial biofilms
Polymer self-healing films containing fragments of pillar [5] arene were obtained for the first
time using thiol/disulfide redox cross-linking. These films were characterized by …
time using thiol/disulfide redox cross-linking. These films were characterized by …
Pyrgos[n]cages: Redefining antibacterial strategy against drug resistance
Y Zhang, M Luo, X Shi, A Li, W Zhou, Y Yin, H Wang… - Science …, 2024 - science.org
Amid rising antibiotic resistance, the quest for advanced antibacterial agents to surpass
microbial adaptation is paramount. This study introduces Pyrgos [n] cages (n= 1 to 4) …
microbial adaptation is paramount. This study introduces Pyrgos [n] cages (n= 1 to 4) …