Recent applications of 1, 3-thiazole core structure in the identification of new lead compounds and drug discovery
A Ayati, S Emami, A Asadipour, A Shafiee… - European Journal of …, 2015 - Elsevier
Thiazole is one of the most important scaffolds in heterocyclic chemistry and drug design
and discovery. It is widely found in diverse pharmacologically active substances and in …
and discovery. It is widely found in diverse pharmacologically active substances and in …
Biological importance of structurally diversified chromenes
Compounds incorporating the chromene scaffold are largely present in natural products and
display a wide variety of biological activities. Their low toxicity combined to the broad …
display a wide variety of biological activities. Their low toxicity combined to the broad …
New pyrazole derivatives containing 1, 2, 4-triazoles and benzoxazoles as potent antimicrobial and analgesic agents
Azole class of compounds are well known for their excellent therapeutic properties. Present
paper describes about the synthesis of three series of new 1, 2, 4-triazole and benzoxazole …
paper describes about the synthesis of three series of new 1, 2, 4-triazole and benzoxazole …
Recent developments in azole compounds as antibacterial and antifungal agents
XM Peng, GX Cai, CH Zhou - Current Topics in Medicinal …, 2013 - ingentaconnect.com
Azole compounds are an important class of nitrogen heterocycles with electron-rich
property. This special structure endows azole-based derivatives easily bind with the …
property. This special structure endows azole-based derivatives easily bind with the …
Hantzsch reaction: synthesis and characterization of some new 1, 4-dihydropyridine derivatives as potent antimicrobial and antioxidant agents
In the present study two new series of Hantzsch 1, 4-dihydropyridine derivatives (1, 4-DHPs)
containing substituted pyrazole moiety (4a–f and 5a–f) were synthesized by the reaction of 3 …
containing substituted pyrazole moiety (4a–f and 5a–f) were synthesized by the reaction of 3 …
Synthesis, characterization and antimicrobial studies of some new pyrazole incorporated imidazole derivatives
In the present study two series of novel imidazole derivatives containing substituted pyrazole
moiety (3a–d and 5a–j) were synthesized. The first series were synthesized by the reaction …
moiety (3a–d and 5a–j) were synthesized. The first series were synthesized by the reaction …
Synthesis and pharmacological evaluation of some novel 2-(5-hydroxy-5-trifluoromethyl-4, 5-dihydropyrazol-1-yl)-4-(coumarin-3-yl) thiazoles
A series of novel 2-(5-hydroxy-5-trifluoromethyl-4, 5-dihydropyrazol-1-yl)-4-(coumarin-3-yl)
thiazoles (6) were synthesized by condensing 3-(2-bromoacetyl) coumarins (4) with various …
thiazoles (6) were synthesized by condensing 3-(2-bromoacetyl) coumarins (4) with various …
Study on the influences of two thiazole flavor ingredients on Cu corrosion caused by chloride ion
S Mo, HQ Luo, NB Li - Journal of colloid and interface science, 2017 - Elsevier
Green corrosion inhibitors are of great benefit to the protection of pipes or tanks in seawater
systems. The properties of the corrosion inhibitor such as toxicity and anticorrosion …
systems. The properties of the corrosion inhibitor such as toxicity and anticorrosion …
[HTML][HTML] Synthesis and in vitro biological evaluation of new pyrazole chalcones and heterocyclic diamides as potential anticancer agents
Synthesis and characterization of new heterocyclic pyrazole chalcones (4a–e) and diamide
(6a–e) derivatives are described. Pyrazole chalcones were synthesized by the reaction of …
(6a–e) derivatives are described. Pyrazole chalcones were synthesized by the reaction of …
[HTML][HTML] Synthesis, characterization and antibacterial activity of some new pyrazole based Schiff bases
In the present study a series of new Schiff bases were synthesized. All the synthesized
compounds were characterized by IR, 1H NMR, mass spectral and elemental analyses …
compounds were characterized by IR, 1H NMR, mass spectral and elemental analyses …