Vinyl azides in organic synthesis: an overview
Among organic azides, vinyl azides have attracted significant attention, because of their
unique properties in organic synthesis, which led to reports of many types of research on this …
unique properties in organic synthesis, which led to reports of many types of research on this …
Recent Advancements in Strategies for the Synthesis of Imidazoles, Thiazoles, Oxazoles, and Benzimidazoles
Nitrogen‐containing heterocycles such as imidazoles, thiazoles, and oxazoles play a
significant role in the fields of biological and pharmaceutical chemistry. These compounds …
significant role in the fields of biological and pharmaceutical chemistry. These compounds …
Selective access to 4-substituted 2-aminothiazoles and 4-substituted 5-thiocyano-2-aminothiazoles from vinyl azides and potassium thiocyanate switched by …
B Chen, S Guo, X Guo, G Zhang, Y Yu - Organic letters, 2015 - ACS Publications
A highly selective construction of 4-substituted 2-aminothiazoles and 4-substituted 5-
thiocyano-2-aminothiazoles, respectively, catalyzed by palladium (II) acetate and promoted …
thiocyano-2-aminothiazoles, respectively, catalyzed by palladium (II) acetate and promoted …
Visible-light-driven synthesis of 4-alkyl/aryl-2-aminothiazoles promoted by in situ generated copper photocatalyst
WL Lei, T Wang, KW Feng, LZ Wu, Q Liu - ACS Catalysis, 2017 - ACS Publications
Room-temperature synthesis of 4-alkyl/aryl-2-aminothiazoles from vinyl azides and
ammonium thiocyanate was accomplished with the aid of copper salts and blue LED …
ammonium thiocyanate was accomplished with the aid of copper salts and blue LED …
The regioselective synthesis of 2, 5-and 4, 5-disubstituted thiazoles via the cyclization of 2-oxo-2-(amino) ethanedithioates with isocyanides
KR Singh, C Santhosh, TR Swaroop… - Organic & Biomolecular …, 2022 - pubs.rsc.org
The regioselective synthesis of 2-(methylthio)-N-aryl/alkylthiazole-5-carboxamides and ethyl-
5-(aryl/alkyl carbamoyl) thiazole-4-carboxylates was carried out via the base-induced …
5-(aryl/alkyl carbamoyl) thiazole-4-carboxylates was carried out via the base-induced …
SARS-CoV-2 Mpro binding profile and drug-likeness of two novel thiazole derivatives: structural elucidation, DFT studies, ADME-T and molecular docking simulations
L Tumakuru Nagarajappa, K Ravi Singh… - Journal of …, 2023 - Taylor & Francis
Two novel thiazole derivatives, ethyl 5-((4-fluorophenyl) carbamoyl)-thiazole-4-carboxylate
(2b) and ethyl 5-(p-tolylcarbamoyl) thiazole-4-carboxylate (6b) have been synthesized, and …
(2b) and ethyl 5-(p-tolylcarbamoyl) thiazole-4-carboxylate (6b) have been synthesized, and …
Design, synthesis and investigation on the structure–activity relationships of N-substituted 2-aminothiazole derivatives as antitubercular agents
Tuberculosis (TB) is one of the deadliest infectious diseases of all times, and its recent
resurgence is a supreme matter of concern. Co-infection with HIV and, in particular, the …
resurgence is a supreme matter of concern. Co-infection with HIV and, in particular, the …
Palladium-metalated porous organic polymers as recyclable catalysts for the chemioselective synthesis of thiazoles from thiobenzamides and isonitriles
W Tong, WH Li, Y He, ZY Mo, HT Tang, HS Wang… - Organic …, 2018 - ACS Publications
Two types of thiazole derivatives are synthesized through a multistep cascade sequence
with Pd-metalated phosphorus-doped porous organic polymers (POPs) as heterogeneous …
with Pd-metalated phosphorus-doped porous organic polymers (POPs) as heterogeneous …
Revealing the macromolecular targets of fragment‐like natural products
T Rodrigues, D Reker, J Kunze… - Angewandte Chemie …, 2015 - Wiley Online Library
Fragment‐like natural products were identified as ligand‐efficient chemical matter for hit‐to‐
lead development and chemical‐probe discovery. Relying on a computational method using …
lead development and chemical‐probe discovery. Relying on a computational method using …
2, 4-Disubstituted thiazoles as multitargated bioactive molecules
Thiazoles are important heterocyclics exhibiting boundaryless biological activities, such as
antibacterial, antifungal, anti-inflammatory, antitumor, antitubercular, antidiabetic, antiviral …
antibacterial, antifungal, anti-inflammatory, antitumor, antitubercular, antidiabetic, antiviral …