Synthesis and antimicrobial activity of some new thiazole, thiophene and pyrazole derivatives containing benzothiazole moiety

S Bondock, W Fadaly, MA Metwally - European journal of medicinal …, 2010 - Elsevier
In an attempt to find a new class of antimicrobial agents, a series of thiazole, thiophene,
pyrazole and other related products containing benzothiazole moiety were prepared via the …

Synthesis and antimicrobial activity of novel 2-thiazolylimino-5-arylidene-4-thiazolidinones

P Vicini, A Geronikaki, K Anastasia, M Incerti… - Bioorganic & medicinal …, 2006 - Elsevier
New 2-thiazolylimino-5-arylidene-4-thiazolidinones (compounds 4a–j), unsubstituted or
carrying hydroxy, methoxy, nitro and chloro groups on the benzene ring, were synthesized …

[PDF][PDF] Recent Developments and Biological Activities of 2-Aminothiazole Derivatives.

ME Khalifa - Acta Chimica Slovenica, 2018 - researchgate.net
Aminothiazole nuclei and their various derivatives have been long used as precursors for
the synthesis of biologically active molecules. As a typical heterocyclic amine, 2 …

Thiadiazole and thiazole derivatives as potential antimicrobial agents

Ц Khamitova, D Berillo, A Lozynskyi… - Mini Reviews in …, 2024 - benthamdirect.com
Background: This review summarizes data on heterocyclic systems with thiadiazole and
thiazole fragments in molecules as promising antimicrobial agents. Introduction: Thiadiazole …

Synthesis of novel inhibitors of α-glucosidase based on the benzothiazole skeleton containing benzohydrazide moiety and their molecular docking studies

M Taha, NH Ismail, S Lalani, MQ Fatmi… - European journal of …, 2015 - Elsevier
In an effort to design and synthesize a new class of α-glucosidase inhibitor, we synthesized
benzothiazole hybrid having benzohydrazide moiety (5). Compound 5 was reacted with …

Synthesis of new S-derivatives of clubbed triazolyl thiazole as anti-Mycobacterium tuberculosis agents

MR Shiradkar, KK Murahari, HR Gangadasu… - Bioorganic & medicinal …, 2007 - Elsevier
In the present study, a series of N-{4-[(4-amino-5-sulfanyl-4H-1, 2, 4-triazol-3-yl) methyl]-1, 3-
thiazol-2-yl}-2-substituted-amide (1a–d) derivatives were synthesized in good yields and …

Synthesis, anticonvulsant activity and 3D-QSAR study of some prop-2-eneamido and 1-acetyl-pyrazolin derivatives of aminobenzothiazole

ND Amnerkar, KP Bhusari - European Journal of Medicinal Chemistry, 2010 - Elsevier
A series of 6-substituted-[3-substituted-prop-2-eneamido] benzothiazole 9–32 and 6-
substituted-2-[(1-acetyl-5-substituted)-2-pyrazolin-3-yl] aminobenzothiazole 33–56 were …

Synthesis of benzimidazolyl-1, 3, 4-oxadiazol-2ylthio-N-phenyl (benzothiazolyl) acetamides as antibacterial, antifungal and antituberculosis agents

RV Patel, PK Patel, P Kumari, DP Rajani… - European journal of …, 2012 - Elsevier
To affiliate multiple bioactivities in a compact heteronuclei, two series of benzimidazole
based 1, 3, 4-oxadiazoles were synthesized and assessed in vitro for their efficacy as …

Synthesis and antimicrobial activity of 1-(4-aryl-2-thiazolyl)-3-(2-thienyl)-5-aryl-2-pyrazoline derivatives

A Özdemir, G Turan-Zitouni, ZA Kaplancıklı… - European Journal of …, 2007 - Elsevier
Several 1-(4-aryl-2-thiazolyl)-3-(2-thienyl)-5-aryl-2-pyrazoline derivatives were synthesized
by reacting substituted 3-(2-thienyl)-5-aryl-1-thiocarbamoyl-2-pyrazolines with phenacyl …

Spectral, XRD, SEM and biological activities of transition metal complexes of polydentate ligands containing thiazole moiety

MA Neelakantan, SS Marriappan, J Dharmaraja… - … Acta Part A: Molecular …, 2008 - Elsevier
Metal complexes of o-vanillidene–2-aminobenzothiazole have been prepared and
characterized by elemental and spectral (vibrational, electronic, 1H NMR and EPR) data as …