Circadian regulation of drug responses: toward sex-specific and personalized chronotherapy

FA Lévi, A Okyar, E Hadadi… - Annual review of …, 2024 - annualreviews.org
Today's challenge for precision medicine involves the integration of the impact of molecular
clocks on drug pharmacokinetics, toxicity, and efficacy toward personalized chronotherapy …

Circadian rhythm and disease: Relationship, new insights, and future perspectives

AR Neves, T Albuquerque, T Quintela… - Journal of cellular …, 2022 - Wiley Online Library
The circadian system is responsible for internal functions and regulation of the organism
according to environmental cues (zeitgebers). Circadian rhythm dysregulation or …

Circadian biology to advance therapeutics for mood disorders

A Bhatnagar, G Murray, S Ray - Trends in Pharmacological Sciences, 2023 - cell.com
Mood disorders account for a significant global disease burden, and pharmacological
innovation is needed as existing medications are suboptimal. A wide range of evidence …

Circadian dysfunction in adipose tissue: chronotherapy in metabolic diseases

E Civelek, D Ozturk Civelek, YK Akyel, D Kaleli Durman… - Biology, 2023 - mdpi.com
Simple Summary The circadian timing system is our bodies' built-in clock and controls our
physiology on a daily basis. This system helps us adapt to changes in our environment, such …

[HTML][HTML] Interactions of circadian clock genes with the hallmarks of cancer

SM Ortega-Campos, EM Verdugo-Sivianes… - … et Biophysica Acta (BBA …, 2023 - Elsevier
The molecular machinery of the circadian clock regulates the expression of many genes and
processes in the organism, allowing the adaptation of cellular activities to the daily light-dark …

Identification of novel small molecules targeting core clock proteins to regulate circadian rhythm

IH Kavakli, S Gul, M Turkay - Current Opinion in Chemical Engineering, 2022 - Elsevier
The circadian rhythms are physiological, biochemical, and behavioral oscillations that cycle
every 24 hours to anticipate the daily changes in the external environment. Disruption of the …

Single nucleotide polymorphisms (SNPs) in circadian genes: Impact on gene function and phenotype

I Baris, O Ozcan, IH Kavakli - Advances in protein chemistry and structural …, 2023 - Elsevier
Circadian rhythm is an endogenous timing system that allows an organism to anticipate and
adapt to daily changes and regulate various physiological variables such as the sleep-wake …

The secondary pocket of cryptochrome 2 is important for the regulation of its stability and localization

GC Parlak, BB Camur, S Gul, O Ozcan, I Baris… - Journal of Biological …, 2022 - ASBMB
Human clock-gene variations contribute to the phenotypic differences observed in various
behavioral and physiological processes, such as diurnal preference, sleep, metabolism …

Why does circadian timing of administration matter for immune checkpoint inhibitors' efficacy?

A Karaboué, PF Innominato, NI Wreglesworth… - British Journal of …, 2024 - nature.com
Background Tolerability and antitumour efficacy of chemotherapy and radiation therapy can
vary largely according to their time of administration along the 24-h time scale, due to the …

Dynamic regulation of the serine loop by distant mutations reveals allostery in cryptochrome1

O Ozcan, S Gul, IH Kavakli - Journal of Biomolecular Structure and …, 2024 - Taylor & Francis
Cryptochromes (CRYs) are essential components of the molecular clock that generates
circadian rhythm. They inhibit BMAL1/CLOCK-driven transcription at the molecular level …