Microwave encounters ionic liquid: synergistic mechanism, synthesis and emerging applications
Z Zhao, H Li, X Gao - Chemical Reviews, 2023 - ACS Publications
Progress in microwave (MW) energy application technology has stimulated remarkable
advances in manufacturing and high-quality applications of ionic liquids (ILs) that are …
advances in manufacturing and high-quality applications of ionic liquids (ILs) that are …
Discovery of new cholesteryl ester transfer protein inhibitors via ligand-based pharmacophore modeling and QSAR analysis followed by synthetic exploration
Cholesteryl ester transfer protein (CETP) is involved in trafficking lipoprotein particles and
neutral lipids between HDL and LDL and therefore is considered a valid target for treating …
neutral lipids between HDL and LDL and therefore is considered a valid target for treating …
High Target Homology Does Not Guarantee Inhibition: Aminothiazoles Emerge as Inhibitors of Plasmodium falciparum
S Johannsen, RM Gierse, A Krüger… - ACS Infectious …, 2024 - ACS Publications
In this study, we identified three novel compound classes with potent activity against
Plasmodium falciparum, the most dangerous human malarial parasite. Resistance of this …
Plasmodium falciparum, the most dangerous human malarial parasite. Resistance of this …
Application of silica gel-supported polyphosphoric acid (PPA/SiO2) as a reusable solid acid catalyst to the synthesis of 3-benzoylisoxazoles and isoxazolines
K Itoh, T Aoyama, H Satoh, Y Fujii, H Sakamaki… - Tetrahedron letters, 2011 - Elsevier
Application of silica gel-supported polyphosphoric acid (PPA/SiO2) as a reusable solid acid
catalyst to the synthesis of 3-benzoylisoxazoles and isoxazolines - ScienceDirect Skip to …
catalyst to the synthesis of 3-benzoylisoxazoles and isoxazolines - ScienceDirect Skip to …
[HTML][HTML] Design, synthesis, and biological evaluation of benzylamino-methanone based cholesteryl ester transfer protein inhibitors
GA Sheikha, R Abu Khalaf, A Melhem, G Albadawi - Molecules, 2010 - mdpi.com
Cholesteryl ester transfer protein (CETP) is a glycoprotein involved in transporting
lipoprotein particles and neutral lipids between high-density lipoprotein (HDL) and low …
lipoprotein particles and neutral lipids between high-density lipoprotein (HDL) and low …
An expedient route to heterocycles through α-arylation of ketones and arylamides by microwave induced thermal S RN 1 reactions
SM Soria-Castro, DA Caminos, AB Penenory - RSC Advances, 2014 - pubs.rsc.org
Microwave irradiation promotes a quick aromatic nucleophilic substitution by a thermally
induced electron transfer process to form new C–C bonds by the coupling of aryl radicals …
induced electron transfer process to form new C–C bonds by the coupling of aryl radicals …
Selective Metal-Free Deoxygenation of Unsymmetrical 1, 2-Dicarbonyl Compounds by Chlorotrimethylsilane and Sodium Iodide
LZ Yuan, D Renko, I Khelifi, O Provot, JD Brion… - Organic …, 2016 - ACS Publications
For the first time, the combination of chlorotrimethylsilane with NaI is used as a selective
reducting system toward 1, 2-diketones. This combination is successfully evaluated with …
reducting system toward 1, 2-diketones. This combination is successfully evaluated with …
Chemoselective generation of acyl phosphates, acylium ion equivalents, from carboxylic acids and an organophosphate ester in the presence of a Brønsted acid
A Sumita, Y Otani, T Ohwada - Chemical Communications, 2017 - pubs.rsc.org
We describe the chemoselective conversion of carboxylic acids to functional aromatic
ketones promoted by a tailored organophosphate ester in the presence of a Brønsted acid …
ketones promoted by a tailored organophosphate ester in the presence of a Brønsted acid …
Dearomative C–C and C–N bond cleavage of 2-arylindoles: transition-metal-free access to 2-aminoarylphenones
S Luo, Z Hu, Q Zhu - Organic Chemistry Frontiers, 2016 - pubs.rsc.org
A transition-metal-free conversion of 2-arylindoles to 2-aminoarylphenones, using
environmentally benign O2 as the sole oxidant, has been developed. This novel oxidative …
environmentally benign O2 as the sole oxidant, has been developed. This novel oxidative …
Silica-supported polyphosphoric acid in the synthesis of 4-substituted tetrahydroisoquinoline derivatives
We report herein an application of an α-amidoalkylation reaction, as an alternative efficient
synthesis of 4-aryl-and 4-methyl-1, 2, 3, 4-tetrahydroisoquinoline derivatives. The amides …
synthesis of 4-aryl-and 4-methyl-1, 2, 3, 4-tetrahydroisoquinoline derivatives. The amides …