Neurodegenerative, inflammatory and neoplastic brain disorders involve neuroinflammatory
reactions, and a biomarker of neuroinflammation would be useful for diagnostic, drug …

A new and efficient copper-catalyzed C3 aryl-and heteroarylselenation of indoles employing
selenium powder has been developed. The advantages of this chemistry involve the use of …

Mild conditions have been developed to achieve Pd (OAc) 2-catalyzed regioselective cross-
coupling between indoles and potassium aryltrifluoroarylborates in the presence of Cu …

An efficient synthesis of indolo [1, 2-c] quinazoline derivatives has been developed by
copper-catalyzed sequential Ullmann N-arylation and aerobic oxidative C–H amination. The …

The rapid and efficient direct C2‐arylation of free (NH)‐indoles with arylsulfinic acids
proceeded through a microwave‐accelerated palladium‐catalyzed desulfitation reaction. By …

A highly efficient protocol of copper catalysis for the one-pot synthesis of fused dibenzo [b,
f][1, 4] oxazepines is reported. The transformation involves a Smiles rearrangement, leading …

A novel and efficient palladium‐catalyzed C2 arylation of N‐substituted indoles with 1‐
aryltriazenes for the synthesis of 2‐arylindoles was developed. In the presence of BF3⋅ …

Abstract SSR180575 (7‐chloro‐N, N, 5‐trimethyl‐4‐oxo‐3‐phenyl‐3, 5‐dihydro‐4H‐
pyridazino [4, 5‐b] indole‐1‐acetamide) is the lead compound of an original …

In the present study, we considered various pharmacophore hypotheses for TSPO ligands
and an optimal one was selected on the basis of 3D‐QSAR studies. This hypothesis was …

The first example of mono Suzuki-Miyaura cross-coupling of N-Boc-2, 5-dibromopyrrole with
a boronic acid (indol-2-ylboronic acid) is reported. The resulting 2-indolyl-5-bromopyrrole …