The conversion of aryl halides to phenols under mild reaction conditions is a longstanding
and formidable challenge in organic chemistry. Herein, we report the rational design of a …

Parallel synthesis and mass-directed purification of a modular ligand library, high-
throughput experimentation, and rational ligand evolution have led to a novel copper …

A method for the hydroxylation of aryl and heteroaryl halides, promoted by a catalyst based
on a biarylphosphine ligand t BuBrettPhos (L5) and its corresponding palladium precatalyst …

A high-yielding and practical method for the synthesis of phenols from electron-deficient
haloarenes and heteroarenes has been developed. The products are formed from …

In this paper, novel amide linked 1, 2, 3-triazoles containing aryloxy derivatives (8a–l) are
synthesized via copper-catalyzed one-pot sequential hydroxylation-O-alkylation/click …