Nuclear EGFR as a molecular target in cancer

TM Brand, M Iida, N Luthar, MM Starr… - Radiotherapy and …, 2013 - Elsevier
The epidermal growth factor receptor (EGFR) has been one of the most targeted receptors in
the field of oncology. While anti-EGFR inhibitors have demonstrated clinical success in …

[HTML][HTML] Control of cell metabolism by the epidermal growth factor receptor

LA Orofiamma, D Vural, CN Antonescu - Biochimica et Biophysica Acta …, 2022 - Elsevier
The epidermal growth factor receptor (EGFR) triggers the activation of many intracellular
signals that control cell proliferation, growth, survival, migration, and differentiation. Given its …

Fisetin inhibits migration and invasion of human cervical cancer cells by down-regulating urokinase plasminogen activator expression through suppressing the p38 …

RH Chou, SC Hsieh, YL Yu, MH Huang, YC Huang… - PloS one, 2013 - journals.plos.org
Fisetin (3, 3', 4', 7-tetrahydroxyflavone), a naturally occurring flavonoid, has been reported to
inhibit proliferation and induce apoptosis in several cancer types. However, its effect on the …

Receptor tyrosine kinases in the nucleus

G Carpenter, HJ Liao - Cold Spring Harbor perspectives …, 2013 - cshperspectives.cshlp.org
To date, 18 distinct receptor tyrosine kinases (RTKs) are reported to be trafficked from the
cell surface to the nucleus in response to ligand binding or heterologous agonist exposure …

NF-κB–driven suppression of FOXO3a contributes to EGFR mutation-independent gefitinib resistance

CF Chiu, YW Chang, KT Kuo… - Proceedings of the …, 2016 - National Acad Sciences
Therapy with epidermal growth factor receptor (EGFR) tyrosine kinase inhibitors (EGFR-
TKIs, such as gefitinib or erlotinib) significantly prolongs survival time for patients with tumors …

Licochalcone A suppresses migration and invasion of human hepatocellular carcinoma cells through downregulation of MKK4/JNK via NF-κB mediated urokinase …

JP Tsai, PC Hsiao, SF Yang, SC Hsieh, DT Bau… - PloS one, 2014 - journals.plos.org
Hepatocellular cell carcinoma (HCC) is one of the most commonly diagnosed cancers
worldwide and in Taiwan. Chemoprevention of cancer with dietary bioactive compounds …

EGFR modulates DNA synthesis and repair through Tyr phosphorylation of histone H4

RH Chou, YN Wang, YH Hsieh, LY Li, W Xia… - Developmental cell, 2014 - cell.com
Posttranslational modifications of histones play fundamental roles in many biological
functions. Specifically, histone H4-K20 methylation is critical for DNA synthesis and repair …

EGFR targeted therapies and radiation: Optimizing efficacy by appropriate drug scheduling and patient selection

KC Cuneo, MK Nyati, D Ray, TS Lawrence - Pharmacology & therapeutics, 2015 - Elsevier
The epidermal growth factor receptor (EGFR) plays an important role in tumor progression
and treatment resistance for many types of malignancies including head and neck …

Targeting the EGFR/PCNA signaling suppresses tumor growth of triple-negative breast cancer cells with cell-penetrating PCNA peptides

YL Yu, RH Chou, JH Liang, WJ Chang, KJ Su… - PLoS …, 2013 - journals.plos.org
Tyrosine 211 (Y211) phosphorylation of proliferation cell nuclear antigen (PCNA) coincides
with pronounced cancer cell proliferation and correlates with poor survival of breast cancer …

The roles of subcellularly located EGFR in autophagy

H Li, L You, J Xie, H Pan, W Han - Cellular signalling, 2017 - Elsevier
The epidermal growth factor receptor (EGFR) is a well-studied receptor-tyrosine kinase that
serves vital roles in regulation of organ development and cancer progression. EGFR not …