[HTML][HTML] Structure-function-guided design of synthetic peptides with anti-infective activity derived from wasp venom

A Boaro, L Ageitos, MDT Torres, EB Blasco… - Cell Reports Physical …, 2023 - cell.com
Antimicrobial peptides (AMPs) derived from natural toxins and venoms offer a promising
alternative source of antibiotics. Here, through structure-function-guided design, we convert …

Macrophage targeting of nitazoxanide-loaded transethosomal gel in cutaneous leishmaniasis

H Khalid, S Batool, F Din, S Khan… - Royal society open …, 2022 - royalsocietypublishing.org
Topical delivery is preferable over systemic delivery for cutaneous leishmaniasis, because
of its easy administration, reduced systemic adverse effects and low cost. Nitazoxanide …

Co-delivery of amphotericin B and pentamidine loaded niosomal gel for the treatment of Cutaneous leishmaniasis

A Anjum, K Shabbir, FU Din, S Shafique, SS Zaidi… - Drug Delivery, 2023 - Taylor & Francis
Topical drug delivery is preferable route over systemic delivery in case of Cutaneous
leishmaniasis (CL). Among the available agents, amphotericin B (AmB) and pentamidine …

Statistically designed dexibuprofen loaded solid lipid nanoparticles for enhanced oral bioavailability

B Imran, F ud Din, Z Ali, A Fatima, MW Khan… - Journal of Drug Delivery …, 2022 - Elsevier
Abstract Dexibuprofen (DBPN), a non-steroidal anti-inflammatory drug (NSAID), exhibit its
action by inhibiting COX enzymes. It belongs to BCS class Ⅱ drugs, owing to its poor …

Development and optimization of imiquimod-loaded nanostructured lipid carriers using a hybrid design of experiments approach

S Kim, S Abdella, F Abid, F Afinjuomo… - International Journal …, 2023 - Taylor & Francis
Background Imiquimod (IMQ) is an immunomodulating drug that is approved for the
treatment of superficial basal cell carcinoma, actinic keratosis, external genital warts and …

Quality by design for sumatriptan loaded nano-ethosomal mucoadhesive gel for the therapeutic management of nitroglycerin induced migraine

U Shafique, F ud Din, S Sohail, S Batool… - International Journal of …, 2023 - Elsevier
Migraine is a progressive neurological condition often accompanied by nausea and
vomiting. Various drugs have recently been used in the treatment of migraine, including …

Statistical optimization of co-loaded rifampicin and pentamidine polymeric nanoparticles for the treatment of cutaneous leishmaniasis

MM Khan, SS Zaidi, FJ Siyal, SU Khan, G Ishrat… - Journal of Drug Delivery …, 2023 - Elsevier
Topical drug delivery against cutaneous leishmaniasis (CL) serves as an effective alternate
approach to improve efficacy and reduce systemic adverse effects. The purpose of this study …

Metformin HCl-loaded transethosomal gel; development, characterization, and antidiabetic potential evaluation in the diabetes-induced rat model

K Nousheen, FU Din, H Jamshaid, R Afza, SU Khan… - Drug Delivery, 2023 - Taylor & Francis
Herein we designed, optimized, and characterized the Metformin Hydrochloride
Transethosomes (MTF-TES) and incorporate them into Chitosan gel to develop Metformin …

Formulation and statistical optimization of letrozole loaded nanotransferosomal gel for tumor targeting

S Imtiaz, S Sohail, F Din, Z Ali, S Batool… - Pharmaceutical …, 2024 - Taylor & Francis
Letrozole (LTZ) is used as first-line treatment for hormone-positive breast cancer (BC) in
postmenopausal women. However, its poor aqueous solubility and permeability have …

Mannosylated imiquimod-terbinafine co-loaded transethosomes for cutaneous leishmaniasis; assessment of its anti-leishmanial potential, in vivo safety and immune …

H Jamshaid, F ud Din, K Nousheen, SU Khan… - Biomaterials …, 2023 - Elsevier
Current treatment options for cutaneous leishmaniasis are associated with myriad limiting
factors including low penetration, poor efficacy, and drug toxicities. Herein, we reported …