Novel quinoline-based thiosemicarbazide derivatives: synthesis, DFT calculations, and investigation of antitubercular, antibacterial, and antifungal activities
E Özcan, SK Vagolu, MG Gündüz… - ACS …, 2023 - ACS Publications
The discovery of new antimicrobial agents as a means of treating drug-resistant microbial
pathogens is of utmost significance to overcome their immense risk to human well-being …
pathogens is of utmost significance to overcome their immense risk to human well-being …
[HTML][HTML] Pd-, Cu-, and Ni-Catalyzed Reactions: A Comprehensive Review of the Efficient Approaches towards the Synthesis of Antibacterial Molecules
A strong synthetic tool for many naturally occurring chemicals, polymers, and
pharmaceutical substances is transition metal-catalyzed synthesis. A serious concern to …
pharmaceutical substances is transition metal-catalyzed synthesis. A serious concern to …
Linking quinoline ring to 5-nitrofuran moiety via sulfonyl hydrazone bridge: Synthesis, structural characterization, DFT studies, and evaluation of antibacterial and …
In the present work, we report the synthesis, structural characterization, and computational
studies of (E)-N'-((5-nitrofuran-2-yl) methylene) quinoline-8-sulfonohydrazide (QNF) as a …
studies of (E)-N'-((5-nitrofuran-2-yl) methylene) quinoline-8-sulfonohydrazide (QNF) as a …
Benzothiazole derivatives as effective α-glucosidase inhibitors: an insight study of structure-activity relationships and molecular targets
Z Khalifa, R Upadhyay, AB Patel - Medicinal Chemistry Research, 2024 - Springer
In treating the major metabolic disorder diabetes mellitus type-2, the α-glucosidase enzyme
inhibitors play an effective role due to their vital capability of polysaccharide hydrolyzation. A …
inhibitors play an effective role due to their vital capability of polysaccharide hydrolyzation. A …
AlCl3-Catalyzed Cascade Reactions of 1,2,3-Trimethoxybenzene and Adipoyl Chloride: Spectroscopic Investigations and Density Functional Theory Studies
Y Çetinkaya, T Artunç, A Menzek - ACS omega, 2022 - ACS Publications
The reaction of 1, 2, 3-trimethoxybenzene with adipoyl chloride in the presence of AlCl3
gave two isomeric cyclopentene derivatives, 1, 6-bis (2, 3, 4-trimethoxyphenyl) hexane-1, 6 …
gave two isomeric cyclopentene derivatives, 1, 6-bis (2, 3, 4-trimethoxyphenyl) hexane-1, 6 …
[HTML][HTML] A tandem strategy for the synthesis of 2-aminobenzothiazoles via manganese catalyzed CS bond formation
T Aneeja, A Chandravarkar, G Anilkumar - Catalysis Communications, 2024 - Elsevier
The first manganese catalyzed tandem methodology for the synthesis of 2-
aminobenzothiazoles from 2-bromophenyl isothiocyanate and differently substituted amines …
aminobenzothiazoles from 2-bromophenyl isothiocyanate and differently substituted amines …
Investigation of cholinesterase and α-glucosidase enzyme activities, and molecular docking and dft studies for 1, 2-disubstituted cyclopentane derivatives with phenyl …
Abstract Six known products (4–9) were prepared from reaction of adipoyl chloride with 1, 2,
3-trimethoxybenzene according to the literature. From (2, 3, 4-trimethoxyphenyl)(2-(2, 3, 4 …
3-trimethoxybenzene according to the literature. From (2, 3, 4-trimethoxyphenyl)(2-(2, 3, 4 …
N-Iodosuccinimide mediated intramolecular oxidative C(sp2)-S bond formation for the synthesis of 2-aminobenzothiazole derivatives
AA Jichkar, IA Opai, NN Karade - Journal of Sulfur Chemistry, 2022 - Taylor & Francis
An extremely efficient synthetic method for the preparation of 2-aminobenzothiazole
derivatives starting from arylthioureas by using N-iodosuccinimide has been reported. This …
derivatives starting from arylthioureas by using N-iodosuccinimide has been reported. This …
Copper catalyzed CN-bond formation and synthesis of Imidazopyridinone derivatives
The formation of the C–N bond is critical because it allows for the incorporation of nitrogen
into organic molecules. Despite significant advances in this area, the formation of the C–N …
into organic molecules. Despite significant advances in this area, the formation of the C–N …