Pyrazoline hybrids as promising anticancer agents: An up-to-date overview
D Matiadis, M Sagnou - International Journal of Molecular Sciences, 2020 - mdpi.com
Pyrazolines are five-membered heterocycles possessing two adjacent nitrogens. They have
attracted significant attention from organic and medicinal chemists due to their potent …
attracted significant attention from organic and medicinal chemists due to their potent …
A systematic review of synthetic tyrosinase inhibitors and their structure-activity relationship
Z Peng, G Wang, QH Zeng, Y Li, H Liu… - Critical Reviews in …, 2022 - Taylor & Francis
Tyrosinase is a copper-containing oxidation enzyme, which is responsible for the production
of melanin. This enzyme is widely distributed in microorganisms, animals and plants, and …
of melanin. This enzyme is widely distributed in microorganisms, animals and plants, and …
In vitro and in silico studies of fluorinated 2, 3‐disubstituted thiazolidinone‐pyrazoles as potential α‐amylase inhibitors and antioxidant agents
As part of our effort to identify potent α‐amylase inhibitors, in the present study, a novel
series of fluorinated thiazolidinone‐pyrazole hybrid molecules were prepared by the …
series of fluorinated thiazolidinone‐pyrazole hybrid molecules were prepared by the …
An efficient ultrasound-assisted CH3COONa catalyzed synthesis of thiazolidinone molecule: theoretical and nonlinear optical evaluations of thiazolidinone-Schiff base …
Chemical synthesis, structural analysis, theoretical calculations and optical properties
exploration of (E)-2-((E)-(4-nitrobenzylidene) hydrazono)-3-phenyl-4-thiazolidinone 7 (C 16 …
exploration of (E)-2-((E)-(4-nitrobenzylidene) hydrazono)-3-phenyl-4-thiazolidinone 7 (C 16 …
Choline chloride-based DES as solvents/catalysts/chemical donors in pharmaceutical synthesis
DES are mixtures of two or more compounds, able to form liquids upon mixing, with lower
freezing points when compared to the individual constituents (eutectic mixtures). This …
freezing points when compared to the individual constituents (eutectic mixtures). This …
A comprehensive survey upon diverse and prolific applications of chitosan-based catalytic systems in one-pot multi-component synthesis of heterocyclic rings
H Mousavi - International Journal of Biological Macromolecules, 2021 - Elsevier
Heterocyclic compounds are among the most prestigious and valuable chemical molecules
with diverse and magnificent applications in various sciences. Due to the remarkable and …
with diverse and magnificent applications in various sciences. Due to the remarkable and …
Novel Bis-Thiazole Derivatives: Synthesis and Potential Cytotoxic Activity Through Apoptosis With Molecular Docking Approaches
A series of bis-thiazoles 5a–g were synthesized from bis-thiosemicarbazone 3 with
hydrazonoyl chlorides 4a–g. Reaction of 3 with two equivalents of α-halocarbonyl …
hydrazonoyl chlorides 4a–g. Reaction of 3 with two equivalents of α-halocarbonyl …
Quinoline‐based thiazolidinone derivatives as potent cytotoxic and apoptosis‐inducing agents through EGFR inhibition
Quinoline‐based thiazolidinone heterocycles exhibited potent activity in the field of cancer
therapy. Hence, ten quinoline‐based thiazolidinone derivatives were evaluated for their …
therapy. Hence, ten quinoline‐based thiazolidinone derivatives were evaluated for their …
Boosting the antimicrobial performance based on new fused spirothiazolidine framework analogs
WI El-Sofany, EM Flefel, OM Darwesh… - Journal of the Iranian …, 2022 - Springer
Abstract New spiro [cyclohexane-1, 2'-thiazolo [4, 5-b] pyridine derivatives (3–23) were
investigated. Then there is in vitro antimicrobial potency against possible organisms …
investigated. Then there is in vitro antimicrobial potency against possible organisms …
[HTML][HTML] New 4-thiazolidinone-based molecules Les-2769 and Les-3266 as possible PPARγ modulators
Abstract Development of cancer drug-resistance is still an ongoing problem in the modern
anticancer treatment. Therefore, there is a need to search for a new active substance, which …
anticancer treatment. Therefore, there is a need to search for a new active substance, which …