A review on the chemistry, coordination, structure and biological properties of 1-(acyl/aroyl)-3-(substituted) thioureas

A Saeed, U Flörke, MF Erben - Journal of Sulfur Chemistry, 2014 - Taylor & Francis
This review provides an overview of the chemistry, structure and potential applications of 1-
(acyl/aroyl)-3-(mono-substituted) and 1-(acyl/aroyl)-3, 3-(di-substituted) thioureas, with …

New naphthoquinone thiazole hybrids as carbonic anhydrase and cholinesterase inhibitors: Synthesis, crystal structure, molecular docking, and acid dissociation …

C Efeoglu, O Selcuk, B Demir, E Sahin, H Sari… - Journal of Molecular …, 2024 - Elsevier
Abstract In this study, N-[3-(3-amino-1, 4-dioxo-1, 4-dihydronaphthalen-2-yl)-4-R-thiazol-2
(3H)-ylidene]-2, 6-difluorobenzamide derivatives as new 1, 4-naphthoquinone thiazole …

Design, synthesis, characterization, and biological evaluation of nicotinoyl thioureas as antimicrobial and antioxidant agents

B Özgeriş - The Journal of Antibiotics, 2021 - nature.com
Addressed herein a series of thioureas starting from various amines and nicotinic acid have
been synthesized. Notably, thiourea based scaffolds are increasingly employed in medicinal …

New acetylphenol-based acyl thioureas broaden the scope of drug candidates for urease inhibition: synthesis, in vitro screening and in silico analysis

U Zahra, S Zaib, A Saeed, M ur Rehman… - International Journal of …, 2022 - Elsevier
Helicobacter pylori urease remains a validated drug target for the eradication of pervasive
chronic stomach infection that leads to severe human health diseases such as gastritis and …

A greener synthetic protocol for the preparation of carbodiimide

AR Ali, H Ghosh, BK Patel - Tetrahedron Letters, 2010 - Elsevier
A new and facile preparation of symmetrical and unsymmetrical 1, 3-diaryl and aryl-alkyl
carbodiimides via a dehydrosulfurisation of their corresponding thioureas is described …

Tandem regioselective synthesis of tetrazoles and related heterocycles using iodine

R Yella, N Khatun, SK Rout, BK Patel - Organic & Biomolecular …, 2011 - pubs.rsc.org
A one-pot, tandem process has been developed for the synthesis of a library of tetrazoles
from aryl isothiocyanates. Condensation of aryl isothiocyanates with ammonia, and aryl …

Cascade Reaction of Tertiary Enaminones, KSCN, and Anilines: Temperature-Controlled Synthesis of 2-Aminothiazoles and 2-Iminothiazoline

L Yuan, J Liu, K Huang, S Wang, Y Jin… - The Journal of Organic …, 2022 - ACS Publications
A one-pot cascade strategy for the synthesis of 2-aminothiazole derivatives by tertiary
enaminones, KSCN, and anilines was developed. By changing the reaction temperature, the …

Synthesis, Glucosidase Inhibition, and In Silico Modeling Analysis of Highly Fluorinated 2-Imino-1, 3-thiazolines in Search of Potent Antidiabetic Agents

L Zahid, S Zaib, A Saeed, HY Alharbi, MS Aljohani… - ACS …, 2024 - ACS Publications
In the present work, 2-imino-1, 3-thiazolines featuring highly fluorinated fragments were
synthesized through a straightforward cyclization of diversely substituted thioureas with 2 …

Intra-and intermolecular C− S bond formation using a single catalytic system: first direct access to arylthiobenzothiazoles

S Murru, H Ghosh, SK Sahoo, BK Patel - Organic Letters, 2009 - ACS Publications
We have for the first time developed two ligand-assisted Cu (I)-catalyzed sequential intra-
and intermolecular S-arylations leading to the direct synthesis of arylthiobenzothiazoles in …

An efficient synthesis of thiazol-2-imine derivatives via a one-pot, three-component reaction

MM Heravi, S Moghimi - Tetrahedron Letters, 2012 - Elsevier
An efficient synthesis of thiazol-2-imine derivatives via a one-pot, three-component reaction -
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