Amylin: pharmacology, physiology, and clinical potential

DL Hay, S Chen, TA Lutz, DG Parkes, JD Roth… - Pharmacological …, 2015 - Elsevier
Amylin is a pancreatic β-cell hormone that produces effects in several different organ
systems. Here, we review the literature in rodents and in humans on amylin research since …

GPCR modulation by RAMPs

DL Hay, DR Poyner, PM Sexton - Pharmacology & therapeutics, 2006 - Elsevier
Our conceptual understanding of the molecular architecture of G-protein coupled receptors
(GPCRs) has transformed over the last decade. Once considered as largely independent …

Fluorescently-labeled fremanezumab is distributed to sensory and autonomic ganglia and the dura but not to the brain of rats with uncompromised blood brain barrier

R Noseda, AJ Schain, A Melo-Carrillo, J Tien… - …, 2020 - journals.sagepub.com
Background The presence of calcitonin gene-related peptide and its receptors in multiple
brain areas and peripheral tissues previously implicated in migraine initiation and its many …

Targeting VIP and PACAP receptor signaling: new insights into designing drugs for the PACAP subfamily of receptors

J Lu, SJ Piper, P Zhao, LJ Miller, D Wootten… - International journal of …, 2022 - mdpi.com
Pituitary Adenylate Cyclase-Activating Peptide (PACAP) and Vasoactive Intestinal Peptide
(VIP) are neuropeptides involved in a diverse array of physiological and pathological …

[HTML][HTML] Amylin brain circuitry

L Boccia, S Gamakharia, B Coester, L Whiting, TA Lutz… - Peptides, 2020 - Elsevier
Amylin is a peptide hormone that is mainly known to be produced by pancreatic β-cells in
response to a meal but amylin is also produced by brain cells in discrete brain areas albeit …

Molecular studies of CGRP and the CGRP family of peptides in the central nervous system

ER Hendrikse, RL Bower, DL Hay, CS Walker - Cephalalgia, 2019 - journals.sagepub.com
Background Calcitonin gene-related peptide is an important target for migraine and other
painful neurovascular conditions. Understanding the normal biological functions of …

CGRP in the trigeminovascular system: a role for CGRP, adrenomedullin and amylin receptors?

CS Walker, DL Hay - British Journal of Pharmacology, 2013 - Wiley Online Library
The neuropeptide calcitonin gene‐related peptide (CGRP) is reported to play an important
role in migraine. It is expressed throughout the trigeminovascular system. Antagonists …

Pathophysiologic and therapeutic implications of adrenomedullin in cardiovascular disorders

T Ishimitsu, H Ono, J Minami, H Matsuoka - Pharmacology & therapeutics, 2006 - Elsevier
Adrenomedullin (AM) is a vasodilator peptide that originally isolated from
pheochromocytoma tissue. However, the mRNA is expressed in the normal adrenal gland …

Immunohistochemical mapping of calcitonin receptors in the adult rat brain

C Becskei, T Riediger, D Zünd, P Wookey, TA Lutz - Brain research, 2004 - Elsevier
Calcitonin receptors (CTR) have previously been identified in specific regions of the rat
central nervous system using in situ hybridization or autoradiography with iodinated ligands …

Expression of adrenomedullin2/intermedin in human brain, heart, and kidney

R Morimoto, F Satoh, O Murakami, K Totsune, T Suzuki… - Peptides, 2007 - Elsevier
Adrenomedullin2/intermedin (AM2/IMD) is a novel member of the calcitonin/calcitonin gene-
related peptide (CGRP) family. In the present study, we developed a specific …