Microwave enhanced synthesis

S Caddick, R Fitzmaurice - Tetrahedron, 2009 - Elsevier
Microwave technology has become very important in synthesis and it is reasonable to assert
that there are now very few areas of synthetic organic chemistry that have not been shown to …

The impact of microwave-assisted organic synthesis in drug discovery

F Mavandadi, Å Pilotti - Drug discovery today, 2006 - Elsevier
Microwave-assisted organic synthesis has revolutionized organic synthesis. Small
molecules can be built in a fraction of the time required by classical thermal methods. As a …

Mo(CO)6-Mediated Carbamoylation of Aryl Halides

W Ren, M Yamane - The Journal of Organic Chemistry, 2010 - ACS Publications
A simple method for the synthesis of amides has been developed by molybdenum-mediated
carbamoylation of aryl halides. Whereas the conventional palladium-catalyzed three …

Radical-Induced Metal and Solvent-Free Cross-Coupling Using TBAI–TBHP: Oxidative Amidation of Aldehydes and Alcohols with N-Chloramines via C–H Activation

TK Achar, P Mal - The Journal of Organic Chemistry, 2015 - ACS Publications
A solvent-free cross-coupling method for oxidative amidation of aldehydes and alcohols via
a metal-free radial pathway has been demonstrated. The proposed methodology uses the …

Microwave-assisted solution-and solid-phase synthesis of 2-amino-4-arylpyrimidine derivatives

M Matloobi, CO Kappe - Journal of combinatorial chemistry, 2007 - ACS Publications
An efficient and rapid microwave-assisted solution-phase method for the synthesis of 2-
amino-4-arylpyrimidine-5-carboxylic acid derivatives has been developed. The five-step …

Comprehensive survey of combinatorial library synthesis: 2004

RE Dolle - Journal of combinatorial chemistry, 2005 - ACS Publications
Comprehensive Survey of Combinatorial Library Synthesis: 2004 | ACS Combinatorial Science
ACS ACS Publications C&EN CAS Find my institution Log In Journal of Combinatorial Chemistry …

Transformation of Contact‐Explosives Primary Amines and Iodine (III) into a Successful Chemical Reaction under Solvent‐Free Ball Milling Conditions

T Kumar Achar, P Mal - Advanced Synthesis & Catalysis, 2015 - Wiley Online Library
Any synthetic transformation using contact‐explosives primary amines and hypervalent
iodine (III)(phenyliodine diacetate) in constrained media (extreme conditions) is practically …

Microwave-assisted preparation of amides using a stable and reusable mesoporous carbonaceous solid acid

R Luque, V Budarin, JH Clark, DJ Macquarrie - Green Chemistry, 2009 - pubs.rsc.org
Microwave-assisted preparation of amides using a stable and reusable mesoporous
carbonaceous solid acid - Green Chemistry (RSC Publishing) DOI:10.1039/B821392P Royal …

Ligand‐Based Virtual Screening, Parallel Solution‐Phase and Microwave‐Assisted Synthesis as Tools to Identify and Synthesize New Inhibitors of Mycobacterium …

F Manetti, M Magnani, D Castagnolo… - ChemMedChem …, 2006 - Wiley Online Library
In an attempt to identify new inhibitors of the growth of Mycobacterium tuberculosis (MTB),
the causative agent of tuberculosis, a procedure for the generation, design, and screening of …

Parallel Solution-Phase and Microwave-Assisted Synthesis of New S-DABO Derivatives Endowed with Subnanomolar Anti-HIV-1 Activity

F Manetti, JA Esté, I Clotet-Codina… - Journal of medicinal …, 2005 - ACS Publications
A simple and efficient methodology for the parallel solution-phase synthesis has been set up
to obtain a series of thiouracils, in turn selectively S-benzylated under microwave irradiation …