Herein, we report a metallaphotoredox catalysis protocol enabling the efficient
dearomatization of indoles utilizing readily available N-quinolyl benzamides under …

Intramolecular hydroarylation of alkenes through hydrogen atom transfer (HAT) represents a
robust method to prepare benzo-fused heterocycles. However, the reported methods have …

Finding highly active molecular scaffold structures is always the key research content of new
pesticide discovery. In the research and development of new pesticides, the discovery of …

Natural products continue to represent a compelling resource for uncovering chemical
scaffolds characterised by significant structural variability and diverse biological activities …

A systematized survey of reviews and monographs published in 2021 on all aspects of
heterocyclic chemistry is given. Methods for the synthesis, reactivity, and practically useful …

Currently, non-proteinogenic α-amino acids (α-AAs) have attracted increasing interest in bio-
and medicinal chemistry. In this context, the first protocol for the asymmetric synthesis of …

We describe a simple and robust procedure for the Rh (III)-catalyzed [4+ 2] cycloaddition of
feedstock gases enabled through C–H activation. A diverse set of 3, 4-dihydroisoquinolones …

Realization of the one-pot Staudinger/aza-Wittig/Castagnoli–Cushman reaction sequence
for a series of azido aldehydes and homophthalic anhydrides is described. The reaction …

We report operationally facile methods for the synthesis of substituted
dihydroisoquinolinones and tetrahydroisoquinolines from readily accessible o-bromobenzyl …

A novel method for the metal-free synthesis of 3, 4-dihydroisoquinolin-1 (2H)-ones and N-
phenyl oxalamides from 1, 2, 3, 4-tetrahydronisoquinoline and N-phenyl glycine derivatives …