Dihydropyrrolo [1, 2-a] pyrazinone rings are a class of heterocycles present in a wide range
of bioactive natural products and analogues thereof. As a direct result of their bioactivity, the …

The fruiting bodies of Ganoderma sinensis are used as food raw materials of marketed
healthcare products. To gain an insight into the chemical and biological profling of G …

The ability of natural and non-natural dipeptides to act as activators of dioxygen in the
absence of metallic cocatalysts is reported here. Proline-derived 2, 5-diketopiperazines …

We describe a cascade reaction that selectively incorporates oxygen into the carbon−
carbon backbone of alkynes using air as the source. The process starts by lithiating readily …

The production of chiral pyrrolodiketopiperazines under organocatalytic conditions
demonstrates the capacity of bicyclic acylpyrrol lactims to perform as pronucleophiles in …

As a result of screening a panel of marine organisms to identify lead molecules for the
stimulation of endochondral bone formation, the calcareous sponge Pericharax heteroraphis …

This study reveals an alternative sequence for the synthesis of compounds that contain the
pyrrolodiketopiperazine structural motif. Starting with a diketopiperazine precursor, a mild …

A novel acid/base‐co‐catalyzed direct intermolecular α‐amination of various cyclic ketones
has been developed for the first time. The reaction employs molecular oxygen as the sole …

A base‐mediated regioselective electrophilic addition of arenediazonium salts at the C3‐
position of tryptamines followed by cyclization provides an efficient entry to C3‐nitrogenated …

We report here that polysubstituted cyclopent-2-enols can be constructed by the one-pot
reaction of doubly activated cyclopropanes and α-EWG substituted acetonitriles under mild …