Recent developments in the synthesis of nitrogen-containing heterocycles through C–H/N–h bond functionalizations and oxidative cyclization
X Liu, Y Huang, X Meng, J Li, D Wang, Y Chen… - Synlett, 2019 - thieme-connect.com
The synthesis and structure of nitrogen-containing heterocycles are fascinating because
these compounds have a great richness of structural, physicochemical, and biological …
these compounds have a great richness of structural, physicochemical, and biological …
1,3-Dipolar Cycloaddition of Nitrile Imine with Carbon Dioxide: Access to 1,3,4-Oxadiazole-2(3H)-ones
CX Guo, WZ Zhang, N Zhang, XB Lu - The Journal of Organic …, 2017 - ACS Publications
Efficient synthesis of 1, 3, 4-oxadiazole-2 (3 H)-one was achieved by CsF/18-crown-6
mediated 1, 3-dipolar cycloaddition of nitrile imine and 2.0 MPa of CO2. CsF/18-crown-6 …
mediated 1, 3-dipolar cycloaddition of nitrile imine and 2.0 MPa of CO2. CsF/18-crown-6 …
Application of N-Acylbenzotriazoles in the Synthesis of 5-Substituted 2-Ethoxy-1,3,4-oxadiazoles as Building Blocks toward 3,5-Disubstituted 1,3,4-Oxadiazol-2(3H) …
S Wet-Osot, W Phakhodee… - The Journal of Organic …, 2017 - ACS Publications
5-Substituted-2-ethoxy-1, 3, 4-oxadiazoles were conveniently prepared through a one-pot
sequential N-acylation/dehydrative cyclization between ethyl carbazate and N …
sequential N-acylation/dehydrative cyclization between ethyl carbazate and N …
Annulation Reactions of In-Situ-Generated N-(Het)aroyldiazenes with Isothiocyanates Leading to 2-Imino-1,3,4-oxadiazolines
Q Zhao, L Ren, J Hou, W Yu, J Chang - Organic letters, 2018 - ACS Publications
A novel annulation reaction of N-(het) aroyldiazenes and isothiocyanates has been
established. This transformation involves a sequential cyclization and desulfurization …
established. This transformation involves a sequential cyclization and desulfurization …
Synthesis of heterocycles by palladium-catalyzed carbonylative reactions
B Gabriele - Advances in Transition-Metal Mediated Heterocyclic …, 2018 - Elsevier
This chapter is intended to give an overview on the recent developments in the field of the
palladium-catalyzed synthesis of carbonylated heterocycles by the direct introduction of …
palladium-catalyzed synthesis of carbonylated heterocycles by the direct introduction of …
Selective N-functionalization of Arylhydrazines with Primary Alcohols and Acids under PPh3/DDQ System
S Shu, M Yu, W Yu, T Wang… - The Journal of Organic …, 2024 - ACS Publications
We present a PPh3/DDQ-mediated regiospecific selective N-functionalization of
arylhydrazines with primary benzylic alcohols and aryl carboxylic acids for the synthesis of N …
arylhydrazines with primary benzylic alcohols and aryl carboxylic acids for the synthesis of N …
KI-catalyzed reactions of aryl hydrazines with α-oxocarboxylic acids in the presence of CO 2: access to 1, 3, 4-oxadiazol-2 (3 H)-ones
N Yang, H Zhang, G Yuan - Organic Chemistry Frontiers, 2019 - pubs.rsc.org
A novel KI-catalyzed synthesis of 1, 3, 4-oxadiazol-2 (3H)-ones from aryl hydrazines, α-
oxocarboxylic acids and CO2 was reported. This process could effectively utilize CO2 from …
oxocarboxylic acids and CO2 was reported. This process could effectively utilize CO2 from …
One-pot synthesis of 1, 3, 4-oxadiazol-2 (3 H)-ones with CO 2 as a C1 synthon promoted by hypoiodite
N Yang, G Yuan - Organic & Biomolecular Chemistry, 2019 - pubs.rsc.org
A convenient and efficient route has been developed to synthesize 1, 3, 4-oxadiazol-2 (3H)-
ones from CO2, hydrazines and aryl or aliphatic aldehydes. Promoted by hypoiodite (IO−) …
ones from CO2, hydrazines and aryl or aliphatic aldehydes. Promoted by hypoiodite (IO−) …
Palladium-Catalyzed Carbonylative Synthesis of Heterocycles
JB Feng, XF Wu - Advances in Heterocyclic Chemistry, 2017 - Elsevier
Palladium-catalyzed carbonylative coupling reactions have been a powerful method in
organic synthesis. The importance and significance have been described abundantly …
organic synthesis. The importance and significance have been described abundantly …
Copper‐catalyzed One‐pot Synthesis of 1, 3, 4‐Oxadiazol‐2 (3H)‐ones Using DMF as the Carbonyl Source
P Jiang, Q Su, K Ablajan… - European Journal of …, 2024 - Wiley Online Library
A series of 1, 3, 4‐oxadiazol‐2 (3H)‐ones were prepared by an efficient copper‐catalyzed
one‐pot reaction of arylhydrazides, arylboronic acids and DMF. Moderate to good yield of 1 …
one‐pot reaction of arylhydrazides, arylboronic acids and DMF. Moderate to good yield of 1 …