Thiazole: A versatile standalone moiety contributing to the development of various drugs and biologically active agents

MF Arshad, A Alam, AA Alshammari, MB Alhazza… - Molecules, 2022 - mdpi.com
For many decades, the thiazole moiety has been an important heterocycle in the world of
chemistry. The thiazole ring consists of sulfur and nitrogen in such a fashion that the pi (π) …

A comprehensive review in current developments of benzothiazole-based molecules in medicinal chemistry

RS Keri, MR Patil, SA Patil, S Budagumpi - European Journal of Medicinal …, 2015 - Elsevier
Benzothiazole (BTA) and its derivatives are the most important heterocyclic compounds,
which are common and integral feature of a variety of natural products and pharmaceutical …

A review of environmental occurrence, fate, exposure, and toxicity of benzothiazoles

C Liao, UJ Kim, K Kannan - Environmental science & technology, 2018 - ACS Publications
Benzothiazole and its derivatives (BTs) are high production volume chemicals that have
been used for several decades in a large number of industrial and consumer products …

An Exploration about the Interaction of Mild Steel with Hydrochloric Acid in the Presence of N-(Benzo[d]thiazole-2-yl)-1-phenylethan-1-imines

B Chugh, AK Singh, S Thakur, B Pani… - The Journal of …, 2019 - ACS Publications
Cost effective inhibition of mild steel corrosion employing eco-friendly materials is a high
priority subject for industries these days. Therefore, in this work, a series of N-(benzo [d] …

Microwave-assisted synthesis–catalytic applications in aqueous media

AK Rathi, MB Gawande, R Zboril, RS Varma - Coordination Chemistry …, 2015 - Elsevier
The development of sustainable methods directed towards the synthesis of molecules is due
to the heightened awareness and recognition of alternative eco-friendly and economical …

Recent advances in the chemistry and biology of benzothiazoles

RK Gill, RK Rawal, J Bariwal - Archiv der Pharmazie, 2015 - Wiley Online Library
Benzothiazole is a privileged heterocyclic scaffold having a benzene ring fused with a five‐
membered thiazole ring. This moiety has attracted considerable attention because of its …

Screening and molecular docking of novel benzothiazole derivatives as potential antimicrobial agents

MA Morsy, EM Ali, M Kandeel, KN Venugopala… - Antibiotics, 2020 - mdpi.com
The burden of antibiotic resistance necessitates a continued search for new antimicrobials.
We evaluated the antimicrobial activities of novel benzothiazoles synthesized by our group …

Therapeutic advancement of benzothiazole derivatives in the last decennial period

S Tariq, P Kamboj, M Amir - Archiv der Pharmazie, 2019 - Wiley Online Library
Benzothiazole, a fused heterocyclic moiety, has attracted synthetic and medicinal chemists
for good reasons. It is a valuable scaffold that possesses diverse biological activities, such …

Importance of fluorine in benzazole compounds

T Al-Harthy, W Zoghaib, R Abdel-Jalil - Molecules, 2020 - mdpi.com
Fluorine-containing heterocycles continue to receive considerable attention due to their
unique properties. In medicinal chemistry, the incorporation of fluorine in small molecules …

Inhibition of quorum sensing-controlled biofilm formation in Pseudomonas aeruginosa by quorum-sensing inhibitors

E Kalaiarasan, K Thirumalaswamy, BN Harish… - Microbial …, 2017 - Elsevier
Antimicrobial therapy against extensively drug-resistant (XDR) P. aeruginosa biofilms is less
efficient compared to the treatment of equal bacterial counts of free-floating planktonic cells …