Computational and artificial intelligence-based methods for antibody development

J Kim, M McFee, Q Fang, O Abdin, PM Kim - Trends in pharmacological …, 2023 - cell.com
Due to their high target specificity and binding affinity, therapeutic antibodies are currently
the largest class of biotherapeutics. The traditional largely empirical antibody development …

Progress and challenges for the machine learning-based design of fit-for-purpose monoclonal antibodies

R Akbar, H Bashour, P Rawat, PA Robert, E Smorodina… - MAbs, 2022 - Taylor & Francis
Although the therapeutic efficacy and commercial success of monoclonal antibodies (mAbs)
are tremendous, the design and discovery of new candidates remain a time and cost …

ABlooper: fast accurate antibody CDR loop structure prediction with accuracy estimation

B Abanades, G Georges, A Bujotzek… - Bioinformatics, 2022 - academic.oup.com
Motivation Antibodies are a key component of the immune system and have been
extensively used as biotherapeutics. Accurate knowledge of their structure is central to …

[HTML][HTML] Advances in computational structure-based antibody design

AM Hummer, B Abanades, CM Deane - Current opinion in structural biology, 2022 - Elsevier
Antibodies are currently the most important class of biotherapeutics and are used to treat
numerous diseases. Recent advances in computational methods are ushering in a new era …

ImmuneBuilder: Deep-Learning models for predicting the structures of immune proteins

B Abanades, WK Wong, F Boyles, G Georges… - Communications …, 2023 - nature.com
Immune receptor proteins play a key role in the immune system and have shown great
promise as biotherapeutics. The structure of these proteins is critical for understanding their …

Machine-designed biotherapeutics: opportunities, feasibility and advantages of deep learning in computational antibody discovery

W Wilman, S Wróbel, W Bielska… - Briefings in …, 2022 - academic.oup.com
Antibodies are versatile molecular binders with an established and growing role as
therapeutics. Computational approaches to developing and designing these molecules are …

[HTML][HTML] Artificial intelligence in pharmaceutical sciences

M Lu, J Yin, Q Zhu, G Lin, M Mou, F Liu, Z Pan, N You… - Engineering, 2023 - Elsevier
Drug discovery and development affects various aspects of human health and dramatically
impacts the pharmaceutical market. However, investments in a new drug often go …

SAbDab in the age of biotherapeutics: updates including SAbDab-nano, the nanobody structure tracker

C Schneider, MIJ Raybould… - Nucleic acids research, 2022 - academic.oup.com
In 2013, we released the Structural Antibody Database (SAbDab), a publicly available
repository of experimentally determined antibody structures. In the interim, the rapid …

Virtual screening algorithms in drug discovery: A review focused on machine and deep learning methods

TA Oliveira, MP Silva, EHB Maia, AM Silva… - Drugs and Drug …, 2023 - mdpi.com
Drug discovery and repositioning are important processes for the pharmaceutical industry.
These processes demand a high investment in resources and are time-consuming. Several …

The RESP AI model accelerates the identification of tight-binding antibodies

J Parkinson, R Hard, W Wang - Nature communications, 2023 - nature.com
High-affinity antibodies are often identified through directed evolution, which may require
many iterations of mutagenesis and selection to find an optimal candidate. Deep learning …