Strengths, weaknesses, opportunities and challenges for long acting injectable therapies: Insights for applications in HIV therapy

A Owen, S Rannard - Advanced drug delivery reviews, 2016 - Elsevier
Advances in solid drug nanoparticle technologies have resulted in a number of long-acting
(LA) formulations with the potential for once monthly or longer administration. Such …

[HTML][HTML] Nanoneuromedicines for degenerative, inflammatory, and infectious nervous system diseases

HE Gendelman, V Anantharam, T Bronich… - … , Biology and Medicine, 2015 - Elsevier
Interest in nanoneuromedicine has grown rapidly due to the immediate need for improved
biomarkers and therapies for psychiatric, developmental, traumatic, inflammatory, infectious …

[HTML][HTML] Sequential LASER ART and CRISPR treatments eliminate HIV-1 in a subset of infected humanized mice

PK Dash, R Kaminski, R Bella, H Su, S Mathews… - Nature …, 2019 - nature.com
Elimination of HIV-1 requires clearance and removal of integrated proviral DNA from
infected cells and tissues. Here, sequential long-acting slow-effective release antiviral …

Transformation of tenofovir into stable ProTide nanocrystals with long-acting pharmacokinetic profiles

DA Cobb, N Smith, S Deodhar, AN Bade… - Nature …, 2021 - nature.com
Abstract Treatment and prevention of human immunodeficiency virus type one (HIV-1)
infection was transformed through widespread use of antiretroviral therapy (ART). However …

Creation of a long-acting nanoformulated dolutegravir

B Sillman, AN Bade, PK Dash, B Bhargavan… - Nature …, 2018 - nature.com
Potent antiretroviral activities and a barrier to viral resistance characterize the human
immunodeficiency virus type one (HIV-1) integrase strand transfer inhibitor dolutegravir …

[HTML][HTML] Creation of a nanoformulated cabotegravir prodrug with improved antiretroviral profiles

T Zhou, H Su, P Dash, Z Lin, BLD Shetty, T Kocher… - Biomaterials, 2018 - Elsevier
Long-acting parenteral (LAP) antiretroviral drugs have generated considerable interest for
treatment and prevention of HIV-1 infection. One new LAP is cabotegravir (CAB), a highly …

Queueing theory model of pentose phosphate pathway

SM Kloska, K Pałczyński, T Marciniak, T Talaśka… - Scientific reports, 2022 - nature.com
Due to its role in maintaining the proper functioning of the cell, the pentose phosphate
pathway (PPP) is one of the most important metabolic pathways. It is responsible for …

Cutting edge strategies for screening of novel anti-HIV drug candidates against HIV infection: a concise overview of cell based assays

SY Gaikwad, P Phatak, A Mukherjee - Heliyon, 2023 - cell.com
Abstract The advent of Highly Active Antiretroviral Therapy has majorly contributed towards
reducing the morbidity and mortality associated with HIV infected people, thus improving the …

The promise of long-acting antiretroviral therapies: from need to manufacture

HE Gendelman, JE McMillan, AN Bade, B Edagwa… - Trends in …, 2019 - cell.com
Antiretroviral therapy has transformed human immunodeficiency virus infections from certain
death to a manageable chronic disease. Achieving strict adherence to drug regimens that …

[HTML][HTML] Anti-retroviral drugs: current state and development in the next decade

X Zhang - Acta pharmaceutica sinica B, 2018 - Elsevier
The pace of discovery of new antiretroviral (ARV) drugs has slowed, although the efficacy
and safety of once-daily fixed dose combinations have been extensively investigated …