IMiD resistance in multiple myeloma: current understanding of the underpinning biology and clinical impact

S Bird, C Pawlyn - Blood, The Journal of the American Society …, 2023 - ashpublications.org
Immunomodulatory agents (IMiDs) are a cornerstone of treatment for patients with multiple
myeloma. IMiDs are used in therapeutic combinations at all stages of disease and are …

Multiple cereblon genetic changes are associated with acquired resistance to lenalidomide or pomalidomide in multiple myeloma

S Gooding, N Ansari-Pour, F Towfic… - Blood, The Journal …, 2021 - ashpublications.org
Emergence of drug resistance to all available therapies is the major challenge to improving
survival in myeloma. Cereblon (CRBN) is the essential binding protein of the widely used …

Pharmacodynamic changes in tumor and immune cells drive Iberdomide's clinical mechanisms of activity in relapsed and refractory Multiple Myeloma

M Amatangelo, E Flynt, N Stong, P Ray… - Cell Reports …, 2024 - cell.com
Iberdomide is a next-generation cereblon (CRBN)-modulating agent in the clinical
development in multiple myeloma (MM). The analysis of biomarker samples from …

Cereblon gene variants and clinical outcome in multiple myeloma patients treated with lenalidomide

PA Huang, SL Beedie, CH Chau, DJ Venzon, S Gere… - Scientific reports, 2019 - nature.com
Abstract Carfilzomib-lenalidomide-dexamethasone (KRd) therapy has yielded promising
results in patients with newly diagnosed multiple myeloma (NDMM). Cereblon (CRBN) is the …

[PDF][PDF] Unravelling the mechanisms of acquired immunomodulatory drug resistance in multiple myeloma

S Bird - 2023 - repository.icr.ac.uk
Immunomodulatory drugs (IMiDs) are a cornerstone of multiple myeloma treatment and
newer cereblon E3 ligase modulating drugs (CELMoDs) are in clinical trials. However, a …