Reductive amination in the synthesis of pharmaceuticals
OI Afanasyev, E Kuchuk, DL Usanov… - Chemical reviews, 2019 - ACS Publications
Reductive amination plays a paramount role in pharmaceutical and medicinal chemistry
owing to its synthetic merits and the ubiquitous presence of amines among biologically …
owing to its synthetic merits and the ubiquitous presence of amines among biologically …
Recent Advances in Organocatalytic Asymmetric Michael Addition Reactions to α, β‐Unsaturated Nitroolefins
T Das, S Mohapatra, NP Mishra, S Nayak… - …, 2021 - Wiley Online Library
An organocatalyzed asymmetric Michael addition reaction has been established as the most
relevant and dynamic research area for the construction of chiral carbon‐carbon and carbon …
relevant and dynamic research area for the construction of chiral carbon‐carbon and carbon …
Catalytic access to succinimide products containing stereogenic quaternary carbons
A Sadiq, TC Nugent - ChemistrySelect, 2020 - Wiley Online Library
Enantioselective α‐branched aldehyde Michael addition to N‐phenylmaleimide resulting in
non‐stereogenic quaternary carbon containing succinimides is common. Here we …
non‐stereogenic quaternary carbon containing succinimides is common. Here we …
Cooperative Catalysis by Boronic Acid-Amine Bifunctionalized Polyacrylonitrile Fibers in Henry Reaction
H Zhang, H Zhang, H Du, J Xiao, M Tao, N Ma… - ACS …, 2023 - ACS Publications
The acid–base pairing and fabrication method was herein employed to construct acid–base
bifunctional heterogeneous catalysts. The boronic acid group was introduced into primary …
bifunctional heterogeneous catalysts. The boronic acid group was introduced into primary …
Recent Advancement on the Organocatalyzed Asymmetric Conjugate Addition using Maleimide as a Potential Substrate
B Jana, M Mondal, S Halder, A Mahata… - Asian Journal of …, 2023 - Wiley Online Library
Abstract Asymmetric organocatalytic 1, 4‐conjugate addition is considered as an effective,
powerful and sustainable method for carbon‐carbon bond formation. The core structure of …
powerful and sustainable method for carbon‐carbon bond formation. The core structure of …
Tunable Approach to Diverse Phenethylamines via Reduction of 5-Aryloxazolidines with Triethylsilane
AA Smorodina, EM Buev, VS Moshkin… - The Journal of …, 2024 - ACS Publications
A rapid pathway for the synthesis of various β-phenethylamines from aromatic aldehydes
has been developed. Initially, a wide range of 5-aryloxazolidines was prepared via the [3+ 2] …
has been developed. Initially, a wide range of 5-aryloxazolidines was prepared via the [3+ 2] …
Design of heterogeneous organocatalyst for the asymmetric Michael addition of aldehydes to maleimides
G Szőllősi, V Kozma - ChemCatChem, 2018 - Wiley Online Library
Asymmetric Michael additions of isobutyraldehyde to maleimides catalyzed by optically pure
diamines and their sulfonamides were investigated to develop heterogeneous chiral …
diamines and their sulfonamides were investigated to develop heterogeneous chiral …
Catalytic Reductive Alkylation of Amines in Batch and Microflow Conditions Using a Silicon-Wafer-Based Palladium Nanocatalyst
T Sato, Y Uozumi, YMA Yamada - ACS omega, 2020 - ACS Publications
We describe the development of the catalytic reductive alkylation of amines with aldehydes
under the atmospheric pressure of H2 using a brush-like silicon-nanostructure-supported …
under the atmospheric pressure of H2 using a brush-like silicon-nanostructure-supported …
Organocatalytic asymmetric Michael/hemiketalization/acyl transfer reaction of 1, 3-propanediones with (E)-2-(2-nitrovinyl) phenols
An organocatalytic asymmetric cascade Michael/hemiketalization/acyl transfer reaction
between (E)-2-(2-nitrovinyl) phenols and 1, 3-propanediones is disclosed. A cinchona …
between (E)-2-(2-nitrovinyl) phenols and 1, 3-propanediones is disclosed. A cinchona …
Synthesis of the diarylindolizidine alkaloid (+)-Fistulopsine B: Application of an organocatalytic Michael addition reaction
NVG Moorthy, SV Pansare - Tetrahedron, 2018 - Elsevier
Synthesis of the diarylindolizidine alkaloid (+)-Fistulopsine B: Application of an organocatalytic
Michael addition reaction - ScienceDirect Skip to main contentSkip to article Elsevier logo …
Michael addition reaction - ScienceDirect Skip to main contentSkip to article Elsevier logo …