Putative purine nucleoside interacting residues in the malaria parasite purine uptake transporter PfENT1 are critical for transporter function

C Dillague, MH Akabas - Plos one, 2023 - journals.plos.org
Malaria remains a major public health threat for billions of people worldwide. Infection with
obligate intracellular, unicellular parasites from the genus Plasmodium causes malaria …

Impact of Field Isolate Identified Nonsynonymous Single Nucleotide Polymorphisms on Plasmodium falciparum Equilibrative Nucleoside Transporter 1 Inhibitor …

Y Sosa, D Egbo, MH Akabas - ACS infectious diseases, 2019 - ACS Publications
Plasmodium falciparum causes the most severe form of malaria and causes approximately
500 000 deaths per year. P. falciparum parasites resistant to current antimalarial treatments …

[HTML][HTML] Nuevas rutas de permeabilidad en Plasmodium falciparum: consideraciones como blanco farmacológico y avances de los potenciales inhibidores

Y Castañeda-Agudelo, A Pabón-Vidal - Actualidades Biológicas, 2021 - scielo.org.co
Con base en la persistencia de los casos de malaria, dados por múltiples razones, entre las
cuales se encuentra la resistencia de Plasmodium falciparum a los antimálaricos …

[图书][B] Antimalarial Drug Development: Characterization and Targeting of the Malaria Parasite Purine Uptake Pathway to Develop Novel Antimalarial Drugs

YD Sosa - 2020 - search.proquest.com
Malaria remains a major public health issue that affects nearly half of the world's population.
Malaria causes approximately 405,000 deaths per year, mainly in pregnant women and …