An energetic and topological approach to understanding the interplay of noncovalent interactions in a series of crystalline spiropyrrolizine compounds

D Tsering, P Dey, KK Kapoor, SK Seth - ACS omega, 2024 - ACS Publications
Synthesis of quinoline-containing spiropyrrolizine was achieved via a 1, 3-dipolar
cycloaddition reaction of azomethine ylide (generated in situ from ninhydrin and l-proline) …

Structure-property relationship in thioxotriaza-spiro derivative: Crystal structure and molecular docking analysis against SARS-CoV-2 main protease

AHU Kumar, KG Vindya, KJ Pampa… - Journal of Molecular …, 2022 - Elsevier
Detailed structural and non-covalent interactions in thioxotriaza-spiroderivative (DZ2) are
investigated by single crystal structure anslysis and computational approaches. Its results …

Experimental and theoretical investigation of conformational states and noncovalent interactions in crystalline sulfonamides with a methoxyphenyl moiety

M Kowalik, J Brzeski, M Gawrońska, K Kazimierczuk… - …, 2021 - pubs.rsc.org
Four sulfonamide derivatives with a methoxyphenyl moiety, namely N-{4-[(2-methoxyphenyl)
sulfamoyl] phenyl} acetamide (1a), N-{4-[(3-methoxyphenyl) sulfamoyl] phenyl} acetamide …

A comprehensive picture of the structures, energies, and bonding in the alanine dimers

J David, S Gómez, D Guerra, D Guerra… - …, 2021 - Wiley Online Library
High level quantum mechanical computations and extensive stochastic searches of the
potential energy surfaces of the Alanine dimers uncover rich and complex structural and …

Exploring the effect of substituents on the supramolecular assemblies built by non-covalent interactions in three closely related 1, 3, 4-oxadiazole-2 (3H)-thione …

LH Al-Wahaibi, V Krishnan, HM Hassan… - Journal of Molecular …, 2024 - Elsevier
Abstract Three closely related 1, 3, 4-oxadiazole-2 (3H)-thione N-Mannich bases were
synthesized and characterized by spectroscopic and single crystal X-ray diffraction methods …

[HTML][HTML] Investigating the intermolecular interactions in the explicitly solvated complexes of lomustine with water and ethanol

EED Okon, H Louis, D Etiese, TO Unimuke… - Chemical Physics …, 2023 - Elsevier
Lomustine is an alkylating chemotherapy drug that is used to treat diverse types of cancer,
including brain tumors, Hodgkin's lymphoma, and non-Hodgkin's lymphoma, which works by …

Spectroscopic, solvation effects and MD simulation of an adamantane-carbohydrazide derivative, a potential antiviral agent

LH Al-Wahaibi, M Abdalla, YS Mary… - Polycyclic Aromatic …, 2023 - Taylor & Francis
The spectroscopic, solvent effects, reactivity and MD simulations of N'-[(1E)-(2, 6-
dichlorophenyl-methylidene] adamantane-1-carbohydrazide (DMC) are reported. Solvation …

Novel Adamantane-Linked Isothiourea Derivatives as Potential Chemotherapeutic Agents: Synthesis, Structural Insights, and Antimicrobial/Anti-Proliferative Profiles

FAM Al-Omary, N Alvarez, LS Al-Rasheed, N Veiga… - ACS …, 2023 - ACS Publications
In this study, two adamantane-linked isothiourea derivatives containing a common 4-
chlorophenyl substituent coupled with 4-nitrobenzyl or 4-bromobenzyl moieties were …

Structural insights and docking analysis of adamantane-linked 1, 2, 4-triazole derivatives as potential 11β-HSD1 inhibitors

DA Osman, MA Macías, LH Al-Wahaibi, NH Al-Shaalan… - Molecules, 2021 - mdpi.com
The solid-state structural analysis and docking studies of three adamantane-linked 1, 2, 4-
triazole derivatives are presented. Crystal structure analyses revealed that compound 2 …

Weak Noncovalent Interactions in Three Closely Related Adamantane-Linked 1, 2, 4-Triazole N-Mannich Bases: Insights from Energy Frameworks, Hirshfeld Surface …

LH Al-Wahaibi, MA Macías, O Blacque, LS Zondagh… - Molecules, 2022 - mdpi.com
Structural analysis and docking studies of three adamantane-linked 1, 2, 4-triazole N-
Mannich bases (1–3) are presented. Compounds 1, 2 and 3 crystallized in the monoclinic P …