Inhibitors of lactate dehydrogenase isoforms and their therapeutic potentials

C Granchi, S Bertini, M Macchia… - Current medicinal …, 2010 - ingentaconnect.com
In many different species, lactate dehydrogenase (LDH) constitutes a major checkpoint of
anaerobic glycolysis, by catalyzing the reduction of pyruvate into lactate. This enzyme has …

Synthesis, characterization, crystal structures, DFT, TD-DFT, molecular docking and DNA binding studies of novel copper (II) and zinc (II) complexes bearing …

H Kargar, R Behjatmanesh-Ardakani, V Torabi… - Polyhedron, 2021 - Elsevier
A novel series of transition metal complexes of Cu (II) and Zn (II), including:[Cu (L 1) 2]:
C1,[Cu (L 2) 2]: C2,[Cu (L 3) 2]: C3,[Cu (L 4) 2]: C4,[Zn (L 1) 2]: Z1,[Zn (L 2) 2]: Z2,[Zn (L 3) 2] …

Warburg effect, lactate dehydrogenase, and radio/chemo-therapy efficacy

MI Koukourakis, A Giatromanolaki - International Journal of …, 2019 - Taylor & Francis
The anaerobic metabolism of glucose by cancer cells, even under well-oxygenated
conditions, has been documented by Otto Warburg as early as 1927. Micro-environmental …

[HTML][HTML] A novel Schiff base derived from the gabapentin drug and copper (II) complex: Synthesis, characterization, interaction with DNA/protein and cytotoxic activity

Z Shokohi-Pour, H Chiniforoshan… - … of Photochemistry and …, 2016 - Elsevier
A novel Schiff base [C 20 H 23 NO 3], has been prepared and characterized using FT-IR, UV–
vis, 1 H NMR spectroscopy, elemental analysis and X-ray crystallography. A copper (II) …

Modulation of antioxidant enzymes, SIRT1 and NF‐κB by resveratrol and nicotinamide in alcohol‐aflatoxin B1‐induced hepatocellular carcinoma

D Rawat, SK Chhonker, RA Naik… - Journal of Biochemical …, 2021 - Wiley Online Library
Hepatocellular carcinoma (HCC) is the fifth most commonly diagnosed cancer worldwide
and is associated with poor prognosis. The current study aimed to assess the therapeutic …

Lactate dehydrogenase 5 expression in squamous cell head and neck cancer relates to prognosis following radical or postoperative radiotherapy

MI Koukourakis, A Giatromanolaki, S Winter, R Leek… - Oncology, 2009 - karger.com
Objectives: We assessed the expression and the prognostic role of lactate dehydrogenase 5
(LDH5, the major LDH isoenzyme involved in anaerobic glycolysis) in patients with …

In vitro DNA interaction, topoisomerase I/II inhibition and cytotoxic properties of polymeric copper (II) complex bridged with perchlorate ion containing N4-type Schiff …

CG Topkaya, T Göktürk, T Hökelek, ES Cetin… - Journal of Molecular …, 2022 - Elsevier
Cu (II) complex containing p-Cl-isonitrosoacetophenone based on N 4-type Schiff base
ligand was synthesized and characterized by elemental analysis, FTIR, 1 H NMR, 13 C NMR …

Chiral halogenated Schiff base compounds: green synthesis, anticancer activity and DNA-binding study

M Ariyaeifar, HA Rudbari, M Sahihi, Z Kazemi… - Journal of Molecular …, 2018 - Elsevier
Eight enantiomerically pure halogenated Schiff base compounds were synthesized by
reaction of halogenated salicylaldehydes with 3-Amino-1, 2-propanediol (R or S) in water as …

Mononuclear silver (I) complexes with 1, 7-phenanthroline as potent inhibitors of Candida growth

ND Savić, S Vojnovic, BĐ Glišić, A Crochet… - European Journal of …, 2018 - Elsevier
Mononuclear silver (I) complexes with 1, 7-phenanthroline (1, 7-phen),[Ag (NO 3-O, O′)(1,
7-phen-N7) 2](1) and [Ag (1, 7-phen-N7) 2] X, X= ClO 4−(2), CF 3 SO 3−(3), BF 4−(4) and …

Phosphatase-like activity, DNA binding, DNA hydrolysis, anticancer and lactate dehydrogenase inhibition activity promoting by a new bis–phenanthroline dicopper (II) …

S Anbu, M Kandaswamy, S Kamalraj… - Dalton …, 2011 - pubs.rsc.org
A new bis-phenanthroline dicopper (II) complex has been synthesized and characterized by
elemental analysis and spectroscopic methods. The molecular structure of the dinuclear Cu …