New oxazolidinone derivatives as antibacterial agents with improved activity

G Poce, G Zappia, GC Porretta, B Botta… - Expert Opinion on …, 2008 - Taylor & Francis
Background: Considerable efforts have been made in order to find new oxazolidinone-
based antibacterial agents with improved biological profile. Objective: The purpose of this …

WCK 4034: A promising oxazolidinone for treating gram positive infections

S Bhawsar, S Pawar, P Deshpande, R Yeole… - Bioorganic & Medicinal …, 2022 - Elsevier
Increased resistance to gram positive infections have highlighted the limitations of currently
available drug treatments including penicillins, macrolides and glycopeptides. As an …

A tandem sulfoxide-elimination–intramolecular sulfenic acid addition approach to spirocyclic scaffolds for compound library synthesis

SE Gątarz - 2023 - etheses.bham.ac.uk
Spirocyclic scaffolds show high importance and popularity in drug discovery due to their
unique properties as drug molecule skeleton and novelty for patentability. Medicinal …

Substituted piperidinophenyl oxazolidinones

VJ Patil, MV Patel, BK Trivedi, DV Dekhane… - US Patent …, 2012 - Google Patents
The present invention relates to oxazolidinones of Formula I and pharmaceutically
acceptable salts, pharmaceutically acceptable solvates or polymorphs thereof. The invention …

Substituted piperidino phenyloxazolidinones

MV Patel, M Phansalkar, VJ Patil… - US Patent …, 2012 - Google Patents
US8217058B2 - Substituted piperidino phenyloxazolidinones - Google Patents US8217058B2
- Substituted piperidino phenyloxazolidinones - Google Patents Substituted piperidino …

[PDF][PDF] Synthese und trägerarme Radiofluorierung von A2A-Adenosin-Rezeptorliganden für die Positronen-Emissions-Tomographie

MAR Skraban - 2017 - juser.fz-juelich.de
Kurzzusammenfassung Der A2A-Adenosin-Rezeptor (A2AAR) spielt im Gehirn eine
wichtige Rolle bei der Regulation von Glutamat und der Freisetzung von Dopamin …

Substituted piperidino phenyloxazolidinones having antimicrobial activity with improved in vivo efficacy

PK Deshpande, MD Sindkhedkar… - US Patent …, 2014 - Google Patents
The present invention provides agents having antimicrobial activity for preventing and
treating infectious diseases. Thus, the present invention provides novel substituted …