Antifungal activity of thiosemicarbazones, bis (thiosemicarbazones), and their metal complexes
Fungi are ubiquitous in nature, and typically cause little or no environmental or pathogenic
damage to their plant, animal, and human hosts. However, a small but growing number of …
damage to their plant, animal, and human hosts. However, a small but growing number of …
A review on development of bio-active thiosemicarbazide derivatives: Recent advances
There has been substantial attention in the expansion of new thiosemicarbazide derivatives
with diverse biological activities in recent years. Therefore, many scientists have prepared …
with diverse biological activities in recent years. Therefore, many scientists have prepared …
Design, synthesis, and characterization of novel iron chelators: Structure− activity relationships of the 2-benzoylpyridine thiosemicarbazone series and their 3 …
DS Kalinowski, Y Yu, PC Sharpe, M Islam… - Journal of medicinal …, 2007 - ACS Publications
Previously, we demonstrated that the potent antiproliferative activity of the di-2-pyridylketone
thiosemicarbazone (DpT) series of Fe chelators was due to their ability to induce Fe …
thiosemicarbazone (DpT) series of Fe chelators was due to their ability to induce Fe …
Synthesis, cytotoxic and antimalarial activities of benzoyl thiosemicarbazone analogs of isoquinoline and related compounds
R Pingaew, S Prachayasittikul, S Ruchirawat - Molecules, 2010 - mdpi.com
Thiosemicarbazone analogs of papaveraldine and related compounds 1–6 were
synthesized and evaluated for cytotoxic and antimalarial activities. The cytotoxic activity was …
synthesized and evaluated for cytotoxic and antimalarial activities. The cytotoxic activity was …
Synthesis crystal structure of 2-methoxybenzoylhydrazones and evaluation of their α-glucosidase and urease inhibition potential
Compounds 1–30 showed varying degree of α-glucosidase inhibition with IC 50 values
ranging between 187 and 420 μ M. Compounds 1, 2, 3, 6, 8, 12, and 4 (IC 50= 187.7±3.05 …
ranging between 187 and 420 μ M. Compounds 1, 2, 3, 6, 8, 12, and 4 (IC 50= 187.7±3.05 …
Structural studies and investigation on the activity of imidazole-derived thiosemicarbazones and hydrazones against crop-related fungi
DC Reis, AAR Despaigne, JGD Silva, NF Silva… - Molecules, 2013 - mdpi.com
New imidazole derived thiosemicarbazones and hydrazones were prepared by
condensation of 4 (5)-imidazole carboxaldehyde, 4-(1 H-imidazole-1-yl) benzaldehyde and …
condensation of 4 (5)-imidazole carboxaldehyde, 4-(1 H-imidazole-1-yl) benzaldehyde and …
A structural chemistry perspective on the antimalarial properties of thiosemicarbazone metal complexes
KL Summers - Mini Reviews in Medicinal Chemistry, 2019 - ingentaconnect.com
Malaria is a potentially life-threatening disease, affecting approx. 214 million people
worldwide. Malaria is caused by a protozoan, Plasmodium falciparum, which is transmitted …
worldwide. Malaria is caused by a protozoan, Plasmodium falciparum, which is transmitted …
Optimized synthesis of new thiosemicarbazide derivatives with tuberculostatic activity
C Popovici, CM Pavel, V Sunel, C Cheptea… - International Journal of …, 2021 - mdpi.com
Original results are presented in the field of research that addresses the extension of the
reaction of residue of acyl-thiosemicarbazide fixation on the structure of 5 …
reaction of residue of acyl-thiosemicarbazide fixation on the structure of 5 …
Phenoxyacetohydrazide Schiff Bases: β-Glucuronidase Inhibitors
Phenoxyacetohydrazide Schiff base analogs 1–28 have been synthesized and their in vitro
β-glucouoronidase inhibition potential studied. Compounds 1 (IC50= 9.20±0.32 µM), 5 …
β-glucouoronidase inhibition potential studied. Compounds 1 (IC50= 9.20±0.32 µM), 5 …
Synthesis, spectroscopic, and antimicrobial studies on bivalent nickel and copper complexes of bis (thiosemicrbazone)
S Chandra, S Raizada, M Tyagi… - Bioinorganic Chemistry …, 2007 - Wiley Online Library
A series of metal complexes of Cu (II) and Ni (II) having the general composition [M (L) X2]
with benzil bis (thiosemicarbazone) has been prepared and characterized by element …
with benzil bis (thiosemicarbazone) has been prepared and characterized by element …