2, 5-Diketopiperazines (2, 5-DKPs) are cyclodipeptides obtained by the condensation of two
α-amino acids. They not only abound in nature but are often produced as degradation …

Indoles are a significant heterocyclic system in natural products and drugs. They are
important types of molecules and natural products and play a main role in cell biology. The …

Herein, we report the first examples of the synthesis of pyrroloindolines by means of (3+ 2)
dearomative annulation reactions between 3-substituted indoles and highly reactive …

Iron (II) bromide catalyzes the transformation of ortho-substituted aryl azides into 2, 3-
disubstituted indoles through a tandem ethereal C–H bond amination [1, 2]-shift reaction …

Functionalized benzothiophenes are important scaffolds found in molecules with wide
ranging biological activity and in organic materials. We describe an efficient, metal‐free …

Exposure of aromatic carboxamides 1e− 1m, heteroaromatic carboxamides 1n− 1p, and α, β-
unsaturated carboxamides 1q− 1s to 1, 1-dimethylallene in the presence of the a cationic …

Simple indole alkaloids and those with a nonrearranged monoterpenoid unit - Natural Product
Reports (RSC Publishing) DOI:10.1039/B820693G Royal Society of Chemistry View PDF …

A practical and efficient synthesis of C (3)-trifluoromethanesulfanylated hexahydropyrrolo [2,
3-b] indoles 5 from tryptamine derivatives was described. The features of this synthesis …

Prenylated indole alkaloids have long been targets for total synthesis, since they possess a
broad range of medicinal properties and intriguing architectures.[1] Our interest in this family …

The development of visible-light-mediated synthesis of pyrroloindolines via an amidyl
radical cyclization–carbon radical functionalization cascade is reported. The transformation …