International union of basic and clinical pharmacology. XCVIII. Histamine receptors

P Panula, PL Chazot, M Cowart, R Gutzmer… - Pharmacological …, 2015 - ASPET
Histamine is a developmentally highly conserved autacoid found in most vertebrate tissues.
Its physiological functions are mediated by four 7-transmembrane G protein–coupled …

The physiology of brain histamine

RE Brown, DR Stevens, HL Haas - Progress in neurobiology, 2001 - Elsevier
Histamine-releasing neurons are located exclusively in the TM of the hypothalamus, from
where they project to practically all brain regions, with ventral areas (hypothalamus, basal …

International Union of Pharmacology. XIII. Classification of histamine receptors

SJ Hill, CR Ganellin, H Timmerman, JC Schwartz… - Pharmacological …, 1997 - ASPET
The classification of histamine receptors has to date been based on rigorous classical
pharmacological analysis, and as yet, the classification of the three histamine receptors that …

The histamine H3 receptor: structure, pharmacology, and function

G Nieto-Alamilla, R Márquez-Gómez… - Molecular …, 2016 - ASPET
Among the four G protein–coupled receptors (H1–H4) identified as mediators of the biologic
effects of histamine, the H3 receptor (H3R) is distinguished for its almost exclusive …

Cloning and functional expression of the human histamine H3 receptor

TW Lovenberg, BL Roland, SJ Wilson, X Jiang… - Molecular …, 1999 - ASPET
Histamine regulates neurotransmitter release in the central and peripheral nervous systems
through H3 presynaptic receptors. The existence of the histamine H3 receptor was …

Histaminergic transmission in the mammalian brain

JC Schwartz, JM Arrang, M Garbarg… - Physiological …, 1991 - journals.physiology.org
The recognition of histamine (HA)[or 2 (4-imidazolyl) ethylamine] as a messenger molecule
in cell-to-cell communication began early in this century. The early history of HA was …

Comparative anatomy of the histaminergic and other aminergic systems in zebrafish (Danio rerio)

JAN Kaslin, P Panula - Journal of Comparative Neurology, 2001 - Wiley Online Library
The histaminergic system and its relationships to the other aminergic transmitter systems in
the brain of the zebrafish were studied by using confocal microscopy and …

5-HT receptor regulation of neurotransmitter release

KB Fink, M Göthert - Pharmacological reviews, 2007 - ASPET
Serotoninergic neurons in the central nervous system impinge on many other neurons and
modulate their neurotransmitter release. This review focuses on 1) the function of …

The histamine H3 receptor: an attractive target for the treatment of cognitive disorders

TA Esbenshade, KE Browman… - British journal of …, 2008 - Wiley Online Library
The histamine H3 receptor, first described in 1983 as a histamine autoreceptor and later
shown to also function as a heteroreceptor that regulates the release of other …

Histamine inhibits dopamine release in the mouse striatum via presynaptic H3 receptors

E Schlicker, K Fink, M Detzner, M Göthert - Journal of Neural Transmission …, 1993 - Springer
In superfused mouse striatal slices preincubated with [3 H] dopamine 25 nmol/l, the
electrically (3 Hz) evoked tritium overflow was inhibited by histamine 10 μmol/l by 18%. The …