Synthesis and anticancer activity evaluation of some novel imidazo[1,2-a]pyridine based heterocycles containing S-alkyl/aryl moiety

B Kaya, L Yurttaş, M Baysal… - … , Sulfur, and Silicon …, 2024 - Taylor & Francis
Here we report the synthesis and anticancer activities of fourteen novel imidazo [1, 2-a]
pyridine derivatives (6a-6n) containing S-alkyl/aryl moiety. The target compounds were …

Design, synthesis, in vitro antiproliferative evaluation, and kinase inhibitory effects of a new series of imidazo [2, 1-b] thiazole derivatives

MS Abdel-Maksoud, MR Kim, MI El-Gamal… - European journal of …, 2015 - Elsevier
Abstract Design and synthesis of a new series of 5, 6-diarylimidazo [2, 1-b] thiazole
derivatives possessing terminal aryl sulfonamide moiety are described. Their in vitro …

Design, synthesis and biological evaluation of amide derivatives of isoxazole-imidazo [1, 2-a] pyridine as anticancer agents

PK Jami, SR Battula, J Sandhya, UD Parimi - Chemical Data Collections, 2023 - Elsevier
A new series of amide derivatives of isoxazole-imidazo [1, 2-a] pyridine (11a-j) derivatives
have been synthesized and their structures were characterized by analytical data. Further …

Design, synthesis and anticancer activity of sulfenylated imidazo-fused heterocycles

R Chitrakar, D Rawat, R Sistla, LN Vadithe… - Bioorganic & Medicinal …, 2021 - Elsevier
We report herein, the design, synthesis and study of anticancer properties of sulfenylated 2-
phenylimidazo [1, 2-a] pyridines and their analogues. A set of twenty sulfenylated imidazo [1 …

Synthesis of 3-N-/O-/S-methyl-imidazo [1, 2-a] pyridine derivatives for caspase-3 mediated apoptosis induced anticancer activity

D Singh, T Yodun, G Kumar, JA Tali, H Tiwari… - Bioorganic …, 2022 - Elsevier
A library of 49 analogs of imidazo [1, 2-a] pyridine with 2-halo, aryl, styryl and phenylethynyl-
substitution at C-2 position and N-/O-/S-methyl linkage at C-3 position, have been …

Design, synthesis, anticancer activity, and in silico studies of novel imidazo[1,2‐a]pyridine based 1H‐1,2,3‐triazole derivatives

S Endoori, KC Gulipalli, S Bodige… - Journal of …, 2021 - Wiley Online Library
A novel series of imidazo [1, 2‐a] pyridine based 1 H‐1, 2, 3‐triazole derivatives were
designed, synthesized, and evaluated for their anticancer activity against two different …

Iodine catalyzed synthesis of imidazo [1, 2-a] pyrazine and imidazo [1, 2-a] pyridine derivatives and their anticancer activity

R Krishnamoorthy, P Anaikutti - RSC advances, 2023 - pubs.rsc.org
An efficient iodine-catalyzed method for synthesizing imidazo [1, 2-a] pyrazines and imidazo
[1, 2-a] pyridines via one-pot three-component condensations has been reported. The …

Design, synthesis, and biological evaluation of amide derivatives of imidazo[2,1-b][1,3,4]thiadiazole as anticancer agents

G Sridhar, S Palle, J Vantikommu… - Synthetic …, 2020 - Taylor & Francis
A new library of amide derivatives of imidazo [2, 1-b][1, 3, 4] thiadiazoles (11a–j) have
designed and synthesized and their structures determined by 1H NMR, 13C NMR, mass and …

Design, synthesis and biological evaluation of imidazopyridine/pyrimidine-chalcone derivatives as potential anticancer agents

A Kamal, JS Reddy, MJ Ramaiah, D Dastagiri… - …, 2010 - pubs.rsc.org
A new series of imidazo [2, 1-b] pyridine/pyrimidine chalcone derivatives were synthesized
and evaluated for their anticancer activity. These chalcone derivatives showed promising …

Design, synthesis and mechanistic studies of novel imidazo [1, 2-a] pyridines as anticancer agents

AS Ismael, NH Amin, MT Elsaadi… - Bioorganic …, 2022 - Elsevier
Herein, the design, synthesis and mechanistic study of five series of imidazo [1, 2-a]
pyridines 8a-d, 9a-f, 11a-c, 12a-d and 14a-d as anticancer agents were discussed. The …