Synthesis, antibacterial, and antiviral evaluation of new heterocycles containing the pyridine moiety

MS Salem, SI Sakr, WM El‐Senousy… - Archiv der …, 2013 - Wiley Online Library
A facile one‐pot four‐component reaction was utilized to construct 2‐oxo‐1, 2‐
dihydropyridine‐3‐carbonitrile as a scaffold for the synthesis of many fused heterocyclic …

[PDF][PDF] Synthesis and antimicrobial evaluation of some new pyridine based heterocycles

ES Darwish, NA Kheder, AM Farag - Heterocycles, 2010 - scholar.cu.edu.eg
A facile and convenient synthesis of pyridine, pyridazine, 2 (3H)-1, 3, 4-thiadiazole and
pyrazole derivatives incorporating a pyridine-2-ylcarboxamido moiety via the versatile …

Synthetic utility of Pyridinium Bromide: synthesis and antimicrobial activity of novel 2, 4, 6‐Trisubstituted pyridines having pyrazole moiety

SM Gomha, KM Dawood - Journal of Heterocyclic Chemistry, 2017 - Wiley Online Library
Fourteen potentially bioactive pyridines, pendant to pyrazole moiety, were synthesized and
evaluated in vitro for their antimicrobial potential. Treatment of 2‐bromo‐1‐(5‐methyl‐1 …

Synthesis and antimicrobial activity of 5-(2-aminothiazol-4-yl)-3, 4-dihydro-4-phenyl pyrimidin-2(1H)-one

KR Lanjewar, AM Rahatgaonkar, MS Chorghade… - 2009 - nopr.niscpr.res.in
A series of hybrid 5-(2-aminothiazol-4-yl)-3, 4-dihydro-4-phenyl pyrimidin-2 (1H)-ones
(ATDPP) are reported. Efficient cyclocondensation of appropriately substituted 5-(2 …

[HTML][HTML] Synthesis and antimicrobial evaluation of new 1, 4-dihydro-4-pyrazolylpyridines and 4-pyrazolylpyridines

O Prakash, K Hussain, R Kumar, D Wadhwa… - Organic and medicinal …, 2011 - Springer
Abstract Background Dialkyl 1, 4-dihydro-2, 6-dimethylpyridine-3, 5-dicarboxylates (1, 4-
DHP) have now been recognized as vital drugs. Some of these derivatives such as …

Design and synthesis of some new thiophene, thienopyrimidine and thienothiadiazine derivatives of antipyrine as potential antimicrobial agents

HM Aly, NM Saleh, HA Elhady - European journal of medicinal chemistry, 2011 - Elsevier
4-acetamide pyrazolone 2 was synthesized by acetylation of 4-amino antipyrine 1 in
excellent yield. 4-acetamide pyrazolone 2 was exploited as a starting material for the …

Synthesis of novel substituted tetrahydropyrimidine derivatives and evaluation of their pharmacological and antimicrobial activities

NFH Mahmoud, EA Ghareeb - Journal of heterocyclic chemistry, 2019 - Wiley Online Library
Tetrahydropyrimidine derivative 1 was employed as intermediate compound, which in turn
was allowed to react with different electrophilic and nucleophilic reagents to synthesize new …

[PDF][PDF] Synthesis and Antimicrobial Evaluation of Some Bis (thioxopyridine), Bis (pyrazolo-(3, 4-b) pyridine), Bis (thieno (2, 3-b) pyridine), Bis (1, 3, 4-thiadiazole) and …

NA Kheder, YN Mabkhot, AM Farag - Heterocycles, 2008 - triggered.edina.clockss.org
Condensation of the N, N'-(ethane-1, 2-diyl) bis (cyanoacetamide)(1) with aromatic
aldehydes gave the corresponding N, N'-(ethane-1, 2-diyl)-bis (2-cyano-3 …

Synthesis and antimicrobial activity of some new heterocycles incorporating the pyrazolopyridine moiety

S Abu‐Melha - Archiv der Pharmazie, 2013 - Wiley Online Library
2‐Cyano‐N‐(4, 6‐dimethyl‐1H‐pyrazolo [3, 4‐b] pyridin‐3‐yl) acetamide (2) was utilized as
key intermediate for the synthesis of some new coumarin 3, pyridine 4, pyrrole 5, thiazole 8 …

Synthesis and antimicrobial screening of some fused heterocyclic pyrroles

MS Mohamed, AE Rashad, MEA Zaki… - Acta Pharmaceutica, 2005 - hrcak.srce.hr
Sažetak Pyrrole derivatives 1a, b were used as precursors for the preparation of pyrrolo [2, 3-
d] pyrimidine derivatives 2a, b-7a, b. Also, the formation and structure of different …