Synthesis of new thiazole derivatives and evaluation of their antimicrobial and cytotoxic activities

S Dawbaa, AE Evren, Z Cantürk… - Phosphorus, Sulfur, and …, 2021 - Taylor & Francis
Abstract Novel 2-heteroaryl-N-[4-(substituted aryl) thiazol-2-yl] propanamide derivatives (7a–
7o) were synthesized and investigated for their antimicrobial activity. Among the tested …

Synthesis and Antimicrobial Activities of Novel Series of 3‐(4‐(2‐substituted thiazol‐4‐yl) phenyl)‐2‐(4‐methyl‐2‐substituted thiazol‐5‐yl) thiazolidin‐4‐one …

SH Shelke, PC Mhaske, S Narkhade… - Journal of …, 2014 - Wiley Online Library
In the present investigation, a novel series of 3‐(4‐(2‐substituted thiazol‐4‐yl) phenyl)‐2‐(4‐
methyl‐2‐substituted thiazol‐5‐yl) thiazolidin‐4‐one derivatives were synthesized by …

Synthesis, characterization and anti-microbial activities of novel thiazole derivatives.

G Saravanan, V Alagarsamy, TGV Pavitra, GC Kumar… - 2010 - cabidigitallibrary.org
In the present study, a novel thiazoles were synthesized by incorporation of pyrazole moiety
at 2nd position of 2-hydrazinyl-N-(4-phenylthiazol-2-yl) acetamide (5) by treating with …

Synthesis and antimicrobial of certain new thiazolidinone, thiazoline, and thiophene derivatives

MA Gouda, MA Berghot, AI Shoeib… - Phosphorus, Sulfur, and …, 2010 - Taylor & Francis
2-Cyano-N-(9, 10-dioxo-9, 10-dihydro-anthracen-2-yl)-acetamide (1) was utilized as a key
intermediate for the synthesis of thiazolidin-4-one 2 and thiocarbamoyl 5 derivatives via …

Synthesis and Antimicrobial Activity of Phenylthioand Benzylsulfonylacetic Acids Based on 2-amino-5-alkyl (arylalkyl)-1, 3, 4-thiadiazoles

SA Serkov, NV Sigai, NN Kostikova, PV Bulatov… - Pharmaceutical …, 2014 - Springer
SYNTHESIS AND ANTIMICROBIAL ACTIVITY OF PHENYLTHIO- AND BENZYLSULFONYLACETIC
ACIDS BASED ON 2-AMINO-5-ALKYL(ARYLALKYL)-1,3,4-THI Page 1 SYNTHESIS AND …

Synthesis and antimicrobial activities of novel series of 1-((4-methyl-2-substituted thiazol-5-yl) methyleneam INO)-2-substituted isothiourea derivatives

SH Shelke, PC Mhaske, P Hande… - Phosphorus, Sulfur, and …, 2013 - Taylor & Francis
A novel series of 1-((4-methyl-2-substituted thiazol-5-yl) methyleneamino)-2-substituted
isothiourea derivatives was synthesized by alkylation of (Z/E)-1-((4-methyl-2-substituted …

Synthesis of some novel 2, 4-disubstituted thiazoles as possible antimicrobial agents

S Wagle, AV Adhikari, NS Kumari - Phosphorus, Sulfur, and Silicon …, 2008 - Taylor & Francis
A series of 4-aryl-2-(3-methyl-7-substituted quinoxaline-2-one-1-yl)-1, 3-thiazoles (6a–l) and
4-substituted alkyl-2-(3-methyl-7-substituted quinoxaline-2-one-1-yl)-1, 3-thiazoles (8a–i) …

Synthesis and antimicrobial activity of some new heterocycles based on 3-methyl-1-phenyl-5-benzene sulfonamido pyrazole

TI El-Emary, N Al-Muaikel… - Phosphorus, Sulfur, and …, 2002 - Taylor & Francis
Treatment of 3-methyl 1-phenyl-5-amino pyrazole 1 with 4-acetyl benzene sulfonyl chloride
in pyridine gave the sulfonamide 2. Condensation of 2 with aromatic aldehydes …

Synthesis of Some New 4-{2-[(Aryl) amino]-1, 3-thiazol4-yl} benzene-1, 2-diols as Possible Antibacterial and Antifungal Agents

B Narayana, BV Ashalatha, KK Vijaya Raj… - … , Sulfur, and Silicon …, 2006 - Taylor & Francis
Some new 4-{2-[(aryl) amino]-1, 3-thiazol-4-yl} benzene-1, 2-diols are prepared and
characterized by spectral analysis. The newly prepared compounds are studied for their …

[HTML][HTML] Synthesis and evaluation of some new thiazolidin-4-one derivatives as potential antimicrobial agents

BA Baviskar, SS Khadabadi, SL Deore - Journal of Chemistry, 2013 - hindawi.com
A new series of N-{4-methyl-5-[4-(4-oxo-2-phenyl (1, 3-thiazolidin-3-yl)]-5-sulfanyl (1, 2, 4-
triazol-3-yl)-1, 3-thiazol-2-yl} acetamide (7a-l) was synthesized in order to determine their …