Studies toward understanding the SAR around the sulfoximine moiety of the sap‐feeding insecticide sulfoxaflor

AM Buysse, BM Nugent, NX Wang… - Pest management …, 2017 - Wiley Online Library
BACKGROUND The discovery of sulfoxaflor (Isoclast™ active) stemmed from a novel
scaffold‐based approach toward identifying bioactive molecules. It exhibits broad‐spectrum …

Functionalized S-perfluorinated sulfoximines: Preparation and evaluation in catalytic processes

TN Le, P Diter, B Pegot, C Bournaud, M Toffano… - Journal of Fluorine …, 2015 - Elsevier
N-substituted S-perfluoroalkylated sulfoximines were synthesized from the NH sulfoximines
either by a copper coupling reaction with aryl halides or by a reaction with electrophilic …

Calcium (II)‐Catalyzed Chemoselective and Regioselective Epoxide Ring Opening with NH Sulfoximines

NS George, M Kosiuha, A Moquette… - European Journal of …, 2022 - Wiley Online Library
We describe herein a versatile methodology for the synthesis of 1, 2‐sulfoximidoyl ethanols
thanks to a Ca (NTf2) 2‐catalyzed epoxide ring‐opening with NH sulfoximines in 2‐MeTHF …

AutoGPA-Based 3D-QSAR Modeling and Molecular Docking Study on Factor Xa Inhibitors as Anticoagulant Agents

FY Guo, QY Yan, K Lin, WY Hong… - MATEC Web of …, 2016 - matec-conferences.org
The three-dimensional-quantitative structure activity relationship (3D-QSAR) studies were
performed on a series of direct factor Xa (FXa) inhibitors using AutoGPA-based modeling …

[PDF][PDF] N-Funktionalisierungen an Sulfoximinen: N-Alkinylierte, N-Tetrafluorpyridylierte und N-Schwefel-funktionalisierte Sulfoximine

H Fergen - d-nb.info
Schwefel übt seit Jahrtausenden eine besondere Faszination auf die Menschheit aus.
Bereits eine der ersten Alchemistinnen, MARIA PROPHETISSA (auch MARIA HEBRAEA …

α-Functionalisation of Cyclic Sulfoximines via Lithiation-Trapping

G Hartley - 2018 - etheses.whiterose.ac.uk
This thesis describes the development of a general synthetic approach for the
diastereoselective synthesis of a wide range of α-functionalised sulfoximines via lithiation …

[引用][C] Chemical characteristics of direct FXa inhibitors registered for atrial fibrillation

A Bridoux, MM Samama, SA Mousa - Ann Cardiol Cardiovasc Med, 2019